BETd-260

Item number	Size	Delivery time	Price
TGM-T14550-1mg	1 mg	7 - 10 business days*	124.00€
TGM-T14550-5mg	5 mg	7 - 10 business days*	310.00€
TGM-T14550-10mg	10 mg	7 - 10 business days*	468.00€
TGM-T14550-25mg	25 mg	7 - 10 business days*	743.00€
TGM-T14550-50mg	50 mg	7 - 10 business days*	-

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Description: BETd-260, a PROTAC linked by a Cereblon ligand and a BET ligand, has an inhibitory... more

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Product information "BETd-260"

Description: BETd-260, a PROTAC linked by a Cereblon ligand and a BET ligand, has an inhibitory effect on BRD4 protein in leukemic cell lines. Target: PROTACs, Epigenetic Reader Domain. Smiles: N(C1=C2C=3C(NC2=NC(C(NCCCCCC4=C5C(C(=O)N(C5)C6C(=O)NC(=O)CC6)=CC=C4)=O)=N1)=CC(=C(OC)C3)C=7C(C)=NOC7C)C=8N(CC)N=C(C8)C9CC9. References: Zhou B, et al. Discovery of a Small-Molecule Degrader of Bromodomain and Extra-Terminal (BET) Proteins with Picomolar Cellular Potencies and Capable of Achieving Tumor Regression. J Med Chem. 2018 Jan 25,61(2):462-481.

Keywords:	ZBC 260
Supplier:	TargetMol
Supplier-Nr:	T14550

Properties

Application:	Protac(R) reagent
MW:	798.89 D
Formula:	C43H46N10O6

Database Information

CAS :	2093388-62-4\| Matching products
KEGG ID :	K11793 \| Matching products

Handling & Safety

Storage:	-20°C
Shipping:	+20°C (International: +4°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

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