Products from TargetMol
TargetMol, based in Boston, Massachusetts, was founded in 2015 and is a drug screening expert in the life science community. The company offers diverse compound libraries, including FDA-approved libraries, and covers a broad spectrum of small molecule compounds such as inhibitors and agonists as well as recombinant proteins and natural products. TargetMol's products are used by researchers worldwide in areas such as cancer research, neurobiology, inflammation, immunology and metabolism.
More information at: www.targetmol.com
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Prucalopride
Item number: TGM-T2542-100mg
Description: Prucalopride (R-93877) is a selective, high-affinity 5-HT4A/4B receptor agonist (Ki: 2.5/8 nM). It has >290-fold selectivity for 5-HT4A/4B receptor than other 5-HT receptor subtypes. Target: 5-HT Receptor. Smiles: COCCCN1CCC(CC1)NC(=O)c1cc(Cl)c(N)c2CCOc12. References: Briejer MR, et al. Eur J Pharmacol,...
| Keywords: | R-93877 |
| Application: | Targets 5-hydroxytryptamine receptor 4 (HTR4) |
| CAS | 179474-81-8 |
| MW: | 367.87 D |
From 30.00€
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Cabazitaxel
Item number: TGM-T2543-1mL
Description: Cabazitaxel (taxoid XRP6258) is a taxane and antineoplastic agent which is currently used in the therapy of castration-resistant metastatic prostate cancer after failure of docetaxel. Target: Autophagy, Microtubule Associated. Smiles:...
| Keywords: | RPR-116258A, XRP6258, taxoid XRP6258, TXD 258 |
| Application: | Targets tubulin beta (TUBB) |
| CAS | 183133-96-2 |
| MW: | 835.93 D |
48.00€
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Bazedoxifene acetate
Item number: TGM-T2544-100mg
Description: Bazedoxifene acetate (WAY-TES 424) is a novel selective estrogen receptor modulator (SERM). Target: Estrogen/progestogen Receptor, Estrogen Receptor/ERR. Smiles: C(=O)(C)O.c1c(cc2c(c1)n(c(c2C)c1ccc(cc1)O)Cc1ccc(cc1)OCCN1CCCCCC1)O. References: Miller CP, et al. J Med Chem, 2001, 44(11), 1654-1657.
| Keywords: | WAY-140424, TSE 424, WAY-TES 424 |
| Application: | Osteoporosis agent, Selective estrogen receptor modulator (SERM) |
| CAS | 198481-33-3 |
| MW: | 530.67 D |
From 38.00€
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Pimozide
Item number: TGM-T2546-1mL
Description: Pimozide (R6238) is a diphenylbutylpiperidine derivative and a dopamine antagonist with the antipsychotic property. Pimozide selectively inhibits type 2 dopaminergic receptors in the central nervous system (CNS), thereby decreasing dopamine neurotransmission and reducing the occurrence of the motor and...
| Keywords: | R6238 |
| Application: | Targets dopamine receptor D2 (DRD2) |
| CAS | 2062-78-4 |
| MW: | 461.55 D |
From 30.00€
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Diflorasone
Item number: TGM-T2548-100mg
Description: Diflorasone is a synthetic glucocorticoid with anti-inflammatory and immunosuppressive properties. Like other glucocorticoids, diflorasone enters the cell by diffusion across the cell membrane and binds to the glucocorticoid receptor (GR) in the cytoplasm. The receptor complex subsequently translocates...
| Application: | Targets glucocorticoid receptor (NR3C1, GR) |
| CAS | 2557-49-5 |
| MW: | 410.45 D |
From 35.00€
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Robenidine hydrochloride
Item number: TGM-T2549-100mg
Description: Robenidine hydrochloride (Robenidine Hydrochoride) is an anticoccidial agent mainly used in poultry. Target: Antibacterial, Parasite, Antibiotic. Smiles: Cl.Clc1ccc(\C=N\NC(=N)N\N=C\c2ccc(Cl)cc2)cc1. References: Yeom H, et al. Arch Pharm Res. 2013 Mar,36(3):359-65.
| Keywords: | Dexium, Robenidine Hydrochoride, Toraxine, Nugatex, Rasexinium |
| Application: | Coccidiostat (for poultry) |
| CAS | 25875-50-7 |
| MW: | 370.66 D |
From 35.00€
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Etofenamate
Item number: TGM-T2553-1mL
Description: Etofenamate is a non-steroidal anti-inflammatory drug (NSAID) used for the treatment of joint and muscular pain. Target: COX. Smiles: N(C1=C(C(OCCOCCO)=O)C=CC=C1)C2=CC(C(F)(F)F)=CC=C2. References: Bender T, et al. Arzneimittelforschung. 2001,51(6):489-92.
| Application: | Targets prostaglandin-endoperoxide synthase 1 [EC:1.14.99.1] (PTGS1, COX1) |
| CAS | 30544-47-9 |
| MW: | 369.33 D |
From 35.00€
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Aclidinium bromide
Item number: TGM-T2555-100mg
Description: Aclidinium bromide (LAS-W 330) is a synthetic anticholinergic agent that is used as an inhalant for treatment of acute bronchospasm due to chronic bronchitis or emphysema. Aclidinium has not been implicated in causing liver enzyme elevations or clinically apparent acute liver injury. Target: AChR....
| Keywords: | LAS 34273, LAS-W 330 |
| Application: | Bronchodilator, Muscarinic acetylcholine receptor antagonist |
| CAS | 320345-99-1 |
| MW: | 564.55 D |
From 32.00€
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JNJ-3534
Item number: TGM-T25557-100mg
Description: JNJ-3534 is an oral active modulator of RORgammat. Target: Others. Smiles: NA
| Keywords: | JNJ3534, JNJ 3534 |
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Cladribine
Item number: TGM-T2558-100mg
Description: Cladribine (2CdA), an adenosine deaminase inhibitor, is utilized in the treatment of lymphoproliferative diseases. Target: Adenosine deaminase, Apoptosis. Smiles: Nc1nc(Cl)nc2n(cnc12)[C@H]1C[C@H](O)[C@@H](CO)O1. References: Ma J, et al. BMC Cancer. 2011, 11, 255.
| Keywords: | 2-Chloro-2'-deoxyadenosine, CldAdo, 2-chlorodeoxyadenosine, 2CdA |
| Application: | Targets ribonucleoside-diphosphate reductase subunit M1 [EC:1.17.4.1] (RRM1) |
| CAS | 4291-63-8 |
| MW: | 285.69 D |
From 33.00€
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Allylestrenol
Item number: TGM-T2559-1mL
Description: Allylestrenol (Gestanin) is a synthetic steroid with progestational activity. Target: Estrogen/progestogen Receptor. Smiles: [H][C@@]12CC[C@@](O)(CC=C)[C@@]1(C)CC[C@]1([H])[C@@]3([H])CCCC=C3CC[C@@]21[H]. References: Madauss KP, et al. Med Res Rev. 2007 May,27(3):374-400.
| Keywords: | Gestanin, Gestanon, Gestanol |
| Application: | Targets progesterone receptor (PGR, NR3C3) |
| CAS | 432-60-0 |
| MW: | 300.48 D |
29.00€
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Hesperetin
Item number: TGM-T2565-100mg
Description: Hesperetin belongs to the flavanone class of flavonoids. Hesperetin, in the form of its glycoside hesperidin, is the predominant flavonoid in lemons and oranges. Target: Autophagy, p38 MAPK, Apoptosis, 5-HT Receptor, TGF-beta/Smad. Smiles: O=C1C=2C(O[C@@H](C1)C3=CC(O)=C(OC)C=C3)=CC(O)=CC2O....
| CAS | 520-33-2 |
| MW: | 302.28 D |
From 37.00€
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