Products from TargetMol
TargetMol, based in Boston, Massachusetts, was founded in 2015 and is a drug screening expert in the life science community. The company offers diverse compound libraries, including FDA-approved libraries, and covers a broad spectrum of small molecule compounds such as inhibitors and agonists as well as recombinant proteins and natural products. TargetMol's products are used by researchers worldwide in areas such as cancer research, neurobiology, inflammation, immunology and metabolism.
More information at: www.targetmol.com
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5-HT2A&5-HT2C agonist-1
Item number: TGM-T79806-50mg
Description: 5-HT2A&5-HT2C agonist-1 (Example 2) is a dual-acting agent targeting 5-HT2A and 5-HT2C receptors with IC50 values of 196 nM and 0.9 nM, respectively. It is applicable in studying central nervous system disorders, including depression, alcoholism, tobacco and cocaine addiction, inflammation, cluster...
| CAS | 1640-02-4 |
| MW: | 232.32 D |
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JAK kinase-IN-1
Item number: TGM-T79807-50mg
Description: JAK kinase-IN-1 (Example 1) is a potent inhibitor targeting the JAK family, including TYK2, JAK1, JAK2, and JAK3, with IC50 values of 4.2 nM, 32 nM, 27 nM, and 3473 nM, respectively [1]. Target: JAK
| CAS | 2698389-43-2 |
| MW: | 407.44 D |
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KRAS G12C inhibitor 61
Item number: TGM-T79808-50mg
Description: KRAS G12C inhibitor 61 (Example 3) demonstrates potent activity by inhibiting phospho-ERK 1/2 in MIA PaCa-2 cells, with an IC50 value of 9 nM, and is applicable in the research of pancreatic, colorectal, and lung cancers [1]. Target: ERK
| Application: | KRAS G12C inhibitor |
| CAS | 2300967-40-0 |
| MW: | 590.09 D |
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ROCK-IN-8
Item number: TGM-T79809-50mg
Description: ROCK-IN-8 (Example 4), a ROCK inhibitor, exhibits anti-inflammatory properties and is suitable for respiratory and gastro-intestinal disease research, demonstrating an IC50 value below 100 nM [1]. Target: ROCK
| CAS | 1621103-79-4 |
| MW: | 556.61 D |
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Porcn-IN-2
Item number: TGM-T79810-50mg
Description: Porcn-IN-2 (Example 107) is a potent Wnt pathway inhibitor with an IC50 of 0.05 nM, applicable in cancer research including sarcoma, melanoma, skin cancer, hematological tumors, lymphoma, carcinoma, and leukemia [1]. Target: Others
| CAS | 1900754-65-5 |
| MW: | 462.43 D |
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DDR1/2 inhibitor-2
Item number: TGM-T79811-50mg
Description: DDR1/2 Inhibitor-2 (Example 31) serves as an inhibitor of DDR1/DDR2, exhibiting IC50 values below 100 nM. It is applicable in cancer and fibrotic disease research [1]. Target: Others
| Application: | DDR1/2 inhibitor |
| CAS | 2908756-11-4 |
| MW: | 492.45 D |
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Raf inhibitor 3
Item number: TGM-T79813-50mg
Description: Raf inhibitor 3 (Example 30), a potent inhibitor of both B-Raf and C-Raf, exhibits IC50 values below 15 nM. It is applicable in cancer research studies [1]. Target: Raf
| Application: | Raf inhibitor |
| CAS | 1662682-11-2 |
| MW: | 430.46 D |
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pan-KRAS-IN-3
Item number: TGM-T79814-50mg
Description: Pan-KRAS-IN-3 (Example 84) is a pan-KRAS inhibitor suitable for cancer research [1]. Target: Ras
| CAS | 2875116-29-1 |
| MW: | 587.63 D |
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c-Fms-IN-14
Item number: TGM-T79815-50mg
Description: c-Fms-IN-14 (Example 76) is a potent c-Fms kinase inhibitor with an IC50 of 4 nM, used in cancer and autoimmune disease research [1]. Target: c-Fms
| CAS | 1898210-99-5 |
| MW: | 436.51 D |
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S1P1 agonist 6 hemicalcium
Item number: TGM-T79817-50mg
Description: Compound I (S1P1 agonist 6 hemicalcium) is an S1P1 agonist that diminishes autoimmune activity by inhibiting lymphocyte trafficking, and serves as an immunosuppressive agent in researching a range of autoimmune diseases [1]. Target: LPL Receptor
| CAS | 2941310-03-6 |
| MW: | 465.51 D |
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PROTAC BRD4 Degrader-21
Item number: TGM-T79818-50mg
Description: PROTAC BRD4 Degrader-21 (Comp 74), a potent BRD4 degrader, has shown significant inhibition of tumor growth in mouse xenograft models, indicating its potential for anticancer research [1]. Target: Epigenetic Reader Domain
| CAS | 2503036-46-0 |
| MW: | 925.97 D |
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AMB639752
Item number: TGM-T79819-50mg
Description: AMB639752 is a potent inhibitor of diacylglycerol kinase alpha (DGKalpha) that reinstates restimulation-induced cell death (RICD) in SAP-deficient lymphocytes through DGKalpha inhibition within intact cells. This compound is applicable in the research of X-linked lymphoproliferative disease 1 (XLP-1)...
| CAS | 371210-26-3 |
| MW: | 365.43 D |
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