Products from TargetMol
TargetMol, based in Boston, Massachusetts, was founded in 2015 and is a drug screening expert in the life science community. The company offers diverse compound libraries, including FDA-approved libraries, and covers a broad spectrum of small molecule compounds such as inhibitors and agonists as well as recombinant proteins and natural products. TargetMol's products are used by researchers worldwide in areas such as cancer research, neurobiology, inflammation, immunology and metabolism.
More information at: www.targetmol.com
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7-Methoxy obtusifolin
Item number: TGM-T75613-50mg
Description: 7-Methoxy obtusifolin (Compound 4) is a competitive inhibitor of tyrosinase with an inhibitory concentration (IC50) of 7.0 µM [1]. Target: Others
| CAS | 1820806-09-4 |
| MW: | 314.29 D |
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Kouitchenside G
Item number: TGM-T75614-50mg
Description: Kouitchenside G, a natural compound extracted from Swertia kouitchensis, demonstrates inhibitory activity against alpha-Glucosidase, showcasing an IC 50 value of 956 µM [1]. Target: Others
| CAS | 1444411-75-9 |
| MW: | 596.53 D |
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TNIK&MAP4K4-IN-1
Item number: TGM-T79794-50mg
Description: TNIK&MAP4K4-IN-1 (compound A-39) is a potent dual inhibitor of TNIK and MAP4K4/HGK, with IC50 values of 1.29 nM and <10 nM, respectively, in human hepatic stellate cell LX-2, and is applicable in cancer and fibrosis inhibition [1]. Target: Others
| CAS | 2478592-86-6 |
| MW: | 446.47 D |
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USP1-IN-5
Item number: TGM-T79795-50mg
Description: USP1-IN-5 (compound 10) is a potent inhibitor of USP1, with an IC50 of less than 50 nM, and of MDA-MB-436 cells, exhibiting an IC50 of less than 50 nM [1]. Target: Others
| CAS | 2925547-94-8 |
| MW: | 532.52 D |
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USP1-IN-6
Item number: TGM-T79796-50mg
Description: USP1-IN-6 (Compound 11) functions as a potent USP1 inhibitor, exhibiting an IC50 value of less than 50 nM. Additionally, it demonstrates inhibitory activity against MDA-MB-436 cells with a comparable IC50. [1]. Target: Others
| CAS | 2925547-95-9 |
| MW: | 560.57 D |
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PHD-IN-1
Item number: TGM-T79797-50mg
Description: PHD-IN-1 (compound 80) is a potent PHD2 inhibitor with an IC50 value of =5 nM and demonstrates EC50 values of 2.5 µM in EPO Elisa assays in both Caco2-HIF1a-HiBiT-clone-1 and Hep3B cell lines [1]. Target: HIF/HIF Prolyl-Hydroxylase
| CAS | 2924182-31-8 |
| MW: | 441.49 D |
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PHD-IN-2
Item number: TGM-T79798-50mg
Description: PHD-IN-2 (Compound 91), a potent PHD antagonist with an IC50 of less than 5 nM, effectively stimulates erythropoietin synthesis in HEP3B cells with an EC50 of less than 2.5 µM. It is applicable for research purposes across various medical fields, including cardiovascular, metabolic, hematological,...
| CAS | 2924182-42-1 |
| MW: | 501.54 D |
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pan-KRAS-IN-4
Item number: TGM-T79799-50mg
Description: Pan-KRAS-IN-4 (compound 5) is a potent KRAS inhibitor, demonstrating IC50 values of 0.37 nM for Kras G12C and 0.19 nM for Kras G12V [1]. Target: Ras
| CAS | 2885961-55-5 |
| MW: | 636.69 D |
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pan-KRAS-IN-2
Item number: TGM-T79800-50mg
Description: Pan-KRAS-IN-2 (compound 6) is a broad-spectrum KRAS inhibitor exhibiting potent activity with IC50 values of =10 nM against KRAS wild type and its mutants (G12D, G12C, G12V, G12S, G12A, Q61H), while showing significantly reduced inhibition, with an IC50 >10 µM, for the KRAS G13D mutant [1]. Target: Ras....
| CAS | 2882825-14-9 |
| MW: | 584.66 D |
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5-HT2C agonist-3
Item number: TGM-T79802-50mg
Description: 5-HT2C agonist-3 ((+)-19), a selective 5-HT2C agonist (EC50: 24 nM, Ki: 78 nM), exhibits antipsychotic-like activity by blocking amphetamine-induced hyperactivity [1]. Target: 5-HT Receptor
| CAS | 2104810-18-4 |
| MW: | 351.84 D |
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5-HT2C agonist-3 free base
Item number: TGM-T79803-50mg
Description: 5-HT2C agonist-3 ((+)-19) free base is a selective 5-HT2C agonist (EC50: 24 nM, Ki: 78 nM) that exhibits antipsychotic drug-like activity and inhibits Amphetamine-induced hyperactivity [1]. Target: 5-HT Receptor
| CAS | 2104810-17-3 |
| MW: | 315.38 D |
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5-HT2 agonist-1 free base
Item number: TGM-T79805-50mg
Description: Compound 24 (5-HT2 agonist-1 free base) is a potent agonist for 5-HT2A, 5-HT2B, and 5-HT2C receptors, exhibiting IC50 values of 10 nM, 8.3 nM, and 1.6 nM, respectively. It is utilized in research pertaining to depression, alcoholism, tobacco and cocaine addiction, inflammation, cluster headache, PTSD,...
| CAS | 2708279-77-8 |
| MW: | 310.39 D |
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