Products from TargetMol
TargetMol, based in Boston, Massachusetts, was founded in 2015 and is a drug screening expert in the life science community. The company offers diverse compound libraries, including FDA-approved libraries, and covers a broad spectrum of small molecule compounds such as inhibitors and agonists as well as recombinant proteins and natural products. TargetMol's products are used by researchers worldwide in areas such as cancer research, neurobiology, inflammation, immunology and metabolism.
More information at: www.targetmol.com
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Pirinixic Acid
Item number: TGM-T2269-100mg
Description: Pirinixic Acid (NSC 310038) is a synthetic thiacetic acid derivative used in biomedical research, carcinogenic Pirinixic acid is a peroxisome proliferator that activates specific peroxisome proliferator-activated receptors (PPAR). Target: PPAR. Smiles: N(C1=NC(SCC(O)=O)=NC(Cl)=C1)C2=C(C)C(C)=CC=C2....
| Keywords: | Wy-14643, NSC 310038 |
| Application: | PPARalpha activator |
| CAS | 50892-23-4 |
| MW: | 323.8 D |
From 38.00€
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CPCCOEt
Item number: TGM-T22692-100mg
Description: CPCCOEt is a low-affinity, selective, non-competitive, and reversible antagonist of mGluR1b. Target: GluR. Smiles: CCOC(=O)C12CC1\C(=N/O)c1ccccc1O2. References: Litschig S, et al. CPCCOEt, a noncompetitive metabotropic glutamate receptor 1 antagonist, inhibits receptor signaling without affecting...
| Application: | Low affinity, selective, non-competitive mGluR1b antagonist |
| CAS | 179067-99-3 |
| MW: | 247.25 D |
From 46.00€
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Trans-Tranilast
Item number: TGM-T2270-100mg
Description: Trans-Tranilast is an antiallergic drug developed by Kissei Pharmaceuticals. It was approved in 1982 for use in Japan and South Korea for bronchial asthma. Indications for keloid and hypertrophic scar were added in 1993. It has been used for the treatment of allergic disorders such as asthma, allergic...
| Keywords: | Tranilast trans- |
| CAS | 70806-55-2 |
| MW: | 327.33 D |
From 31.00€
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Decloxizine
Item number: TGM-T22713-10mg
Description: Decloxizine is a H1 receptor antagonist. Target: Histamine Receptor. Smiles: Cl.Cl.OCCOCCN1CCN(CC1)C(c1ccccc1)c1ccccc1. References: Farmer LJ, Ledeboer MW, Hoock T, et al. Discovery of VX-509 (Decernotinib): A Potent and Selective Janus Kinase 3 Inhibitor for the Treatment of Autoimmune Diseases. J Med...
| CAS | 3733-63-9 |
| MW: | 340.46 D |
From 33.00€
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BPR1J-097
Item number: TGM-T2272-100mg
Description: BPR1J-097) is a novel FLT-3 inhibitor(IC50: 11±7 nM) with promising in vivo anti-tumor activities. It also inhibits FLT-3 D835Y (IC50: 3 nM). Target: FLT. Smiles: CN1CCN(CC1)c1ccc(cc1)C(=O)Nc1cc([nH]n1)-c1cccc(NS(=O)(=O)c2ccccc2)c1. References: Lin WH, et al. Br J Y. 2012 Jan 31,106(3):475-81.
| Keywords: | BPR1J097 |
| Application: | FLT3 inhibitor |
| CAS | 1327167-19-0 |
| MW: | 516.61 D |
From 48.00€
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Dipsacobioside
Item number: TGM-T22729-1mL
Description: Dipsacobioside is extracted from Anemone hupehensis. Target: Others. Smiles: CC1C(C(C(C(O1)OC2COC(C(C2O)O)OC3CCC4(C(C3(C)CO)CCC5(C4CC=C6C5(CCC7(C6CC(CC7)(C)C)C(=O)O)C)C)C)O)O)O
| CAS | 123350-57-2 |
| MW: | 750.96 D |
From 539.00€
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ITD-1
Item number: TGM-T2273-100mg
Description: ITD-1 is a potent and highly selective TGFbeta pathway inhibitor. Target: TGF-beta/Smad. Smiles: CCOC(=O)C1=C(C)NC2=C(C1c1ccc(cc1)-c1ccccc1)C(=O)CC(C)(C)C2. References: Willems E, et al. Cell Stem Cell. 2012 Aug 3,11(2):242-252.
| Application: | TGF-beta inhibitor, TGF-beta receptor type II degradation inducer |
| CAS | 1099644-42-4 |
| MW: | 415.52 D |
From 32.00€
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DPCPX
Item number: TGM-T22744-10mg
Description: DPCPX (PD 116948) is an A1 adenosine receptor antagonist. Target: Adenosine Receptor. Smiles: C(CC)N1C2=C(NC(=N2)C3CCCC3)C(=O)N(CCC)C1=O. References: Aleksandra S , Ewa P , Karolina B , et al. DPCPX, a selective adenosine A1 receptor antagonist, enhances the antidepressant-like effects of imipramine,...
| Keywords: | PD 116948 |
| Application: | Adenosine A1 receptor antagonist |
| CAS | 102146-07-6 |
| MW: | 304.39 D |
From 39.00€
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Presapogenin CP4
Item number: TGM-T23184-1mL
Description: Presapogenin CP4 extracted from Anemone hupehensis. Target: Others. Smiles: C[C@]12C([C@]3([C@@](C(O)=O)(CC1)CCC(C)(C)C3)[H])=CC[C@]4([C@@]2(C)CC[C@@]5([C@]4(C)CC[C@H](O[C@H]6[C@H](O[C@H]7[C@H](O)[C@H](O[C@H]8[C@H](O)[C@H](O)[C@H](O)CO8)[C@@H](O)[C@H](C)O7)[C@@H](O)[C@@H](O)CO6)C5(C)C)[H])[H]
| CAS | 75799-18-7 |
| MW: | 867.07 D |
From 454.00€
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Indacaterol
Item number: TGM-T2320-1mL
Description: Indacaterol (Onbrez, Arcapta) is a beta2-Adrenergic Agonist. The mechanism of action of indacaterol is as an Adrenergic beta2-Agonist. Target: Adrenergic Receptor. Smiles: CCc1cc2CC(Cc2cc1CC)NC[C@H](O)c1ccc(O)c2[nH]c(=O)ccc12. References: Battram, C., et al., In vitro and in vivo pharmacological...
| Application: | Targets adrenergic receptor beta-2 (ADRB2) |
| CAS | 312753-06-3 |
| MW: | 392.49 D |
From 41.00€
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Quinacrine (dihydrochloride hydrate)
Item number: TGM-T23210-1g
Description: Quinacrine is a compound that is commonly used as an anti-protozoal agent. It inhibits voltage-dependent sodium channels (IC50: 3.3 µM) and suppresses aldehyde oxidase (IC50: 3.3 µM). Quinacrine prevents misfolding of prion protein (EC50: 0.3 µM). As an effective riboflavin antagonist, quinacrine...
| Keywords: | Quinacrine (hydrochloride hydrate) (83-89-6 free base) |
| MW: | 472.9 D |
From 48.00€
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Darunavir
Item number: TGM-T2324-100mg
Description: Darunavir (TMC114) is an HIV PROTEASE INHIBITOR that is used in the treatment of AIDS and HIV INFECTIONS. Due to the emergence of ANTIVIRAL DRUG RESISTANCE when used alone, it is administered in combination with other ANTI-HIV AGENTS. Target: HIV Protease. Smiles:...
| Keywords: | TMC114 |
| Application: | Targets HIV protease [EC:3.4.23.16 3.4.23.47] (PR) |
| CAS | 206361-99-1 |
| MW: | 547.66 D |
From 30.00€
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