Products from TargetMol
TargetMol, based in Boston, Massachusetts, was founded in 2015 and is a drug screening expert in the life science community. The company offers diverse compound libraries, including FDA-approved libraries, and covers a broad spectrum of small molecule compounds such as inhibitors and agonists as well as recombinant proteins and natural products. TargetMol's products are used by researchers worldwide in areas such as cancer research, neurobiology, inflammation, immunology and metabolism.
More information at: www.targetmol.com
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Antitumor agent-75
Item number: TGM-T62510-100mg
Description: Antitumor agent-75 is a novel and potent antitumor agent with cytotoxic effects on both cancer and normal human cell lines. In combination with antitumor agent-74, Antitumor agent-75 exhibits a highly selective cytotoxic effect (IC50: 2.8 µM) against human lung adenocarcinoma [cell line A549]. Antitumor...
| MW: | 438.5 D |
From 1,440.00€
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Imidocarb dihydrochloride monohydrate
Item number: TGM-T62520-100mg
Description: Imidocarb dihydrochloride monohydrate is an effective antiprotozoal agent against the parasite B. bovis (IC50: 87 µg/ml). Target: Others
| MW: | 439.34 D |
From 1,440.00€
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HIV-1 inhibitor-8
Item number: TGM-T62526-100mg
Description: HIV-1 inhibitor-8 is a potent, orally active, low toxicity HIV-1 non-nucleoside reverse transcriptase inhibitor (NNRTI). HIV-1 inhibitor-8 is capable of acting on WT HIV-1 reverse transcriptase (IC50: 0.081 µM). HIV-1 inhibitor-8 exhibited potent antiviral effects against various HIV-1 strains with EC50...
| MW: | 439.53 D |
From 903.00€
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Dopamine D3 receptor ligand-1
Item number: TGM-T62528-100mg
Description: Dopamine D3 receptor ligand is a potent, selective, high-affinity compound with 89 times greater selectivity for D3 receptors (Ki: 8 nM) compared to D2 receptors (Ki: 715 nM). Target: Others
| MW: | 439.55 D |
From 1,440.00€
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Antimalarial agent 7
Item number: TGM-T62537-100mg
Description: Antimalarial agent 7 is a potent and effective inhibitor of PfATP4, showing potential for studying human Plasmodium falciparum. Target: Others
| MW: | 440.44 D |
From 1,440.00€
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PARP1/BRD4-IN-2
Item number: TGM-T62540-100mg
Description: PARP1/BRD4-IN-2 is a potent and selective inhibitor of PARP1 (IC50: 197 nM) and BRD4 (IC50: 238 nM), which inhibits DNA damage repair, blocks the G0/G1 cell cycle transition, and induces apoptosis. PARP1/BRD4-IN-2 exhibits antitumor effects in the MDA-MB-468 mouse xenograft tumor model and is used to...
| MW: | 440.45 D |
From 1,440.00€
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AChE-IN-22
Item number: TGM-T62541-100mg
Description: AChE-IN-22 (compound 10q) is a selective acetylcholinesterase (AChE) inhibitor with IC50 values of 0.88 µM for AChE and 10 µM for BuChE. It binds to both the catalytic active site (CAS) and peripheral anionic site (PAS) of AChE and is used in Alzheimer's disease research. Target: Others
| MW: | 440.47 D |
From 1,440.00€
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DSM705 hydrochloride
Item number: TGM-T62550-100mg
Description: DSM705 hydrochloride is a potent antimalarial compound and a pyrrole-based inhibitor of dihydroorotate dehydrogenase (DHODH).DSM705 hydrochloride shows nanomolar effects against PlasmodiumDHODH and Plasmodium parasites and does not inhibit mammalian DHODH. Target: Others
| MW: | 440.85 D |
From 1,127.00€
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PPARgamma phosphorylation inhibitor 1
Item number: TGM-T62554-100mg
Description: PPARgamma phosphorylation inhibitor 1 (Compound 10) is a potent PPARgamma binding agent (IC50: 24 nM) with antidiabetic effects, inhibiting CDK5-mediated PPARgamma Ser273 phosphorylation (IC50: 160 nM) and displaying minimal PPARgamma agonism. Target: Others
| MW: | 441.26 D |
From 1,440.00€
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JAK-IN-23
Item number: TGM-T62556-100mg
Description: JAK-IN-23 is an orally active dual JAK/STAT and NF-kappaB inhibitor that inhibits JAK1 (IC50: 8.9 nM), JAK2 (IC50: 15 nM), and JAK3 (IC50: 46.2 nM). It exhibits strong anti-inflammatory effects and can reduce the release of various pro-inflammatory factors. JAK-IN-23 can be used to study inflammatory...
| MW: | 441.35 D |
From 867.00€
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Mu opioid receptor antagonist 5
Item number: TGM-T62673-100mg
Description: Mu opioid receptor antagonist 5 (compound NAP) is a selective mu opioid receptor (MOR) antagonist that crosses the blood-brain barrier, with an EC50 of 1.14 nM and a Ki of 0.37 nM. Mu opioid receptor antagonist 5 can be used to study opioid use disorder (OUD). Target: Others
| MW: | 447.53 D |
From 1,440.00€
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LSD1-IN-21
Item number: TGM-T62674-100mg
Description: LSD1-IN-21 is a potent, blood-brain barrier permeable LSD1 (lysine specific demethylase-1) inhibitor (IC50: 0.956 µM).LSD1-IN-21 significantly reduces the pro-inflammatory cytokine TNF-alpha and exhibits good anti-cancer and anti-inflammatory effects. Target: Others
| MW: | 447.55 D |
From 1,440.00€
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