Products from TargetMol

TargetMol

TargetMol, based in Boston, Massachusetts, was founded in 2015 and is a drug screening expert in the life science community. The company offers diverse compound libraries, including FDA-approved libraries, and covers a broad spectrum of small molecule compounds such as inhibitors and agonists as well as recombinant proteins and natural products. TargetMol's products are used by researchers worldwide in areas such as cancer research, neurobiology, inflammation, immunology and metabolism.

More information at: www.targetmol.com

Go to the catalogs of TargetMol

11563 from 12311 pages
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TrxR-IN-2
TrxR-IN-2

Item number: TGM-T62021-100mg

Description: TrxR-IN-2 is a potential thioredoxin reductase (TrxR) inhibitor. TrxR-IN-2 has research value in the chemotherapy of drug-resistant hepatocellular carcinoma. Target: Others
MW: 406.43 D
From 1,440.00€ *
Review
GSK852
GSK852

Item number: TGM-T62024-100mg

Description: GSK852 is a potent, second bromodomain (BD2)-selective, bromo and extra-terminal domain (BET) inhibitor with pIC50 of 7.9. Target: Others
MW: 406.47 D
From 1,440.00€ *
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GAK inhibitor 49 hydrochloride
GAK inhibitor 49 hydrochloride

Item number: TGM-T62027-100mg

Description: GAK inhibitor 49 hydrochloride is a potent, highly selective, ATP-competitive inhibitor of cyclin G-associated kinase (GAK) with a Ki of 0.54 nM and a cell IC50 of 56 nM. It can also bind to RIPK2. Target: Others
MW: 406.86 D
From 1,051.00€ *
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CDK2-IN-8
CDK2-IN-8

Item number: TGM-T62038-100mg

Description: CDK2-IN-8 is a potent CDK2 inhibitor (IC50 = 1.74 µM) that exhibits antiproliferative activity and can be used for melanoma research. Target: Others
MW: 407.47 D
From 1,440.00€ *
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L-365260 hemihydrate
L-365260 hemihydrate

Item number: TGM-T62039-100mg

Description: L-365260 hemihydrate is a selective, orally active non-peptide gastrin and brain cholecystokinin receptor (CCK-B) antagonist, demonstrating competitive interaction with guinea pig stomach gastrin and brain CCK receptors and exhibiting inhibition constants (Kis) of 1.9 nM and 2.0 nM, respectively....
MW: 407.47 D
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XP5
XP5

Item number: TGM-T62041-100mg

Description: XP5 is a potent, orally active HDAC6 inhibitor (IC50= 31 nM) that inhibits the proliferation of various cancer cell lines, including HDACi-resistant YCC3/7 gastric cancer cells (IC50=0.16-2.31 µM). Target: Others
MW: 407.48 D
From 1,440.00€ *
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Dyrk1A/B-IN-1
Dyrk1A/B-IN-1

Item number: TGM-T62043-100mg

Description: Dyrk1A/B-IN-1 (compound 3n) is a potent, selective, and cell-permeable inhibitor of DYRK1A and DYRK1B, with Kis of 67.8 nM and 237.9 nM, and IC 50 s of 1.1 µM and 0.8 µM, respectively. Target: Others
MW: 407.51 D
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Topo I-IN-1
Topo I-IN-1

Item number: TGM-T62048-100mg

Description: Topo I-IN-1 (Compound 14d) is a potent Topo I inhibitor that exhibits antitumor activity, DNA intercalative capability, and can induce cell apoptosis. Target: Others
MW: 408.25 D
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D4R antagonis-2
D4R antagonis-2

Item number: TGM-T62054-100mg

Description: D4R antagonist-2 is a potent and selective D4R antagonist (IC50= 6.52 µM) with favorable in vitro pharmacokinetic parameters and good brain penetration, making it a potential research candidate for Parkinson's disease. Target: Others
MW: 408.87 D
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Anticancer agent 12
Anticancer agent 12

Item number: TGM-T62057-100mg

Description: Anticancer agent 12 shows cytotoxic activity in malignant cells with no hepatotoxicity. Target: Others
MW: 409.3 D
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MAO-B-IN-7
MAO-B-IN-7

Item number: TGM-T62062-100mg

Description: MAO-B-IN-7 is a potent and blood-brain barrier permeable MAO-B and AChE inhibitor, exhibiting IC50 values of 41 nM for human AChE, 87 nM for electric eel AChE, and 0.3 µM for MAO-B. MAO-B-IN-7 effectively alleviates oxidative stress and neuroinflammatory damage. Target: Others
MW: 409.52 D
From 1,440.00€ *
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Antibacterial agent 76
Antibacterial agent 76

Item number: TGM-T62063-100mg

Description: Antibacterial agent 76 (compound 9) is a potent antibacterial agent. Target: Others
MW: 409.54 D
From 1,440.00€ *
Review
11563 from 12311 pages