Products from TargetMol
TargetMol, based in Boston, Massachusetts, was founded in 2015 and is a drug screening expert in the life science community. The company offers diverse compound libraries, including FDA-approved libraries, and covers a broad spectrum of small molecule compounds such as inhibitors and agonists as well as recombinant proteins and natural products. TargetMol's products are used by researchers worldwide in areas such as cancer research, neurobiology, inflammation, immunology and metabolism.
More information at: www.targetmol.com
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Ziprasidone amino acid
Item number: TGM-T73961-10mg
Description: Ziprasidone amino acid (Ziprasidone Impurity C), an impurity found in Ziprasidone, functions as a combined 5-HT (serotonin) and dopamine receptor antagonist, demonstrating significant antipsychotic activity [1]. Target: Others
| MW: | 430.95 D |
From 198.00€
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Cetirizine Impurity C dihydrochloride
Item number: TGM-T73962-50mg
Description: Cetirizine Impurity C dihydrochloride, a specific impurity of Cetirizine, is associated with a second-generation antihistamine that serves as the carboxylated metabolite of hydroxyzine. This compound acts as a specific, orally active, and long-acting antagonist of the histamine H1-receptor [1] [2]....
| CAS | 2702511-37-1 |
| MW: | 461.81 D |
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Imatinib Impurity E
Item number: TGM-T73973-50mg
Description: Imatinib Impurity E is a specific impurity found in Imatinib, an orally available inhibitor of multiple tyrosine kinases, including BCR/ABL, v-Abl, PDGFR, and c-kit. Imatinib (STI571) operates by semi-competitively inhibiting enzyme activity, it binds adjacent to the ATP binding site, inducing a closed...
| CAS | 1365802-18-1 |
| MW: | 873.02 D |
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(S)-Dehydro Venlafaxine
Item number: TGM-T73977-50mg
Description: (S)-Dehydro Venlafaxine is an inactive S-enantiomer of Dehydro Venlafaxine. Dehydro Venlafaxine is an impurity of Venlafaxine hydrochloride. Venlafaxine hydrochloride (Wy 45030 hydrochloride) is a potent serotonin (5-HT) / norepinephrine (NE) reuptake dual inhibitor [1] [2] . Target: Others
| MW: | 259.39 D |
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Cidofovir diphosphate tri(triethylamine)
Item number: TGM-T73983-50mg
Description: Cidofovir diphosphate triethylamine, an active intracellular metabolite of Cidofovir, acts as a selective inhibitor of viral DNA polymerases. It exhibits inhibitory constants (K_i) of 6.6 µM for human cytomegalovirus (HCMV) DNA polymerase, 0.86 µM for herpes simplex virus-1 (HSV-1) DNA polymerase, and...
| MW: | 742.72 D |
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ONX-0914 TFA
Item number: TGM-T73986-50mg
Description: ONX-0914 (PR-957) TFA is a selective, noncompetitive, irreversible inhibitor of the chymotrypsin-like subunit (LMP7) of the immunoproteasome, effectively blocking cytokine production and mitigating experimental arthritis progression. With a K_i value of 5.2 µM against the mycobacterial proteasome,...
| MW: | 694.7 D |
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Nedosiran sodium
Item number: TGM-T73994-50mg
Description: Nedosiran sodium, a GalNAc-dsRNA conjugate, is engineered to suppress the synthesis of the hepatic lactate dehydrogenase (LDH) enzyme. Target: Others
| Application: | Targets L-lactate dehydrogenase [EC:1.1.1.27] (LDH, ldh) |
| CAS | 2247026-22-6 |
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EGFR/CSC-IN-1
Item number: TGM-T73995-50mg
Description: EGFR/CSC-IN-1 is a dual inhibitor of the epidermal growth factor receptor (EGFR [IC50 10.52 nM]) and cancer stem cells (CSC), potentially applicable in triple-negative breast cancer research. Target: EGFR
| CAS | 2820447-02-5 |
| MW: | 1067.08 D |
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Anti gram-positive/negative bacteria agent 1
Item number: TGM-T73997-50mg
Description: Anti gram-positive/negative bacteria agent 1 is an antibiotic conjugated with a synthetic MECAM-based siderophore, designed to combat both gram-positive and gram-negative bacteria. Target: Others
| MW: | 1381.38 D |
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CP-547632 TFA
Item number: TGM-T74000-100mg
Description: CP-547632 TFA is an orally active, ATP-competitive inhibitor that potently targets VEGFR-2 and FGF kinases with IC50 values of 11 nM and 9 nM, respectively. It demonstrates selectivity for VEGFR-2 and bFGF over EGFR, PDGFRbeta, and related tyrosine kinases (TKs), exhibiting antitumor efficacy [1]....
| CAS | 2805804-54-8 |
| MW: | 646.43 D |
From 1,867.00€
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INY-03-041 trihydrochloride
Item number: TGM-T74001-50mg
Description: INY-03-041 trihydrochloride, a potent and highly selective PROTAC-based pan-AKT degrader, comprises Ipatasertib, an ATP-competitive AKT inhibitor, conjugated to Lenalidomide. It effectively inhibits AKT1, AKT2, and AKT3 with IC50 values of 2.0, 6.8, and 3.5 nM, respectively [1]. Target: PROTACs
| MW: | 907.8 D |
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SJF620 hydrochloride
Item number: TGM-T74002-50mg
Description: SJF620 hydrochloride is a PROTAC that utilizes a lenalidomide analog to recruit CRBN and ligands to target Btk, exhibiting a DC50 of 7.9 nM [1]. Target: PROTACs
| CAS | 2821938-05-8 |
| MW: | 797.3 D |
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