Products from TargetMol
TargetMol, based in Boston, Massachusetts, was founded in 2015 and is a drug screening expert in the life science community. The company offers diverse compound libraries, including FDA-approved libraries, and covers a broad spectrum of small molecule compounds such as inhibitors and agonists as well as recombinant proteins and natural products. TargetMol's products are used by researchers worldwide in areas such as cancer research, neurobiology, inflammation, immunology and metabolism.
More information at: www.targetmol.com
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Anti-MRSA agent 16
Item number: TGM-T88982-10mg
Description: Anti-MRSA agent 16 (Compound 4) acts as an inhibitor against methicillin-resistant Staphylococcus aureus (MRSA). When used in combination with oxacillin or meropenem, it proves effective in treating infected mice. Target: Antibacterial
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E3 Ligase Ligand-linker Conjugate 111
Item number: TGM-T88987-10mg
Description: E3LigaseLigand-linker Conjugate 111 is an E3 ubiquitin ligase ligand-linker conjugate. Target: E3 Ligase Ligand-Linker Conjugate
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PBE-AMF
Item number: TGM-T88991-10mg
Description: PBE-AMF is a prodrug that activates H2O2 and exhibits anticancer activity. It impedes tumor proliferation by inhibiting DNA synthesis, reducing ATP levels, inducing cell death (apoptosis), and blocking the cell cycle. PBE-AMF effectively and selectively inhibits the proliferation of MDA-MB-231 cells...
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PBA-AMF
Item number: TGM-T89007-10mg
Description: PBA-AMF is activated by H2O2, releasing formamide (AMF). This compound selectively inhibits the proliferation of breast cancer cells without affecting non-cancerous cells. It works by inhibiting DNA synthesis, reducing ATP levels, inducing apoptosis (Apoptosis), and arresting the cell cycle, thereby...
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L-703606 oxalate hydrate
Item number: TGM-T89016-10mg
Description: L-703606 oxalate hydrate is an effective, selective NK1 receptor antagonist. It is utilized in research related to gastric acid secretion. Target: Neurokinin receptor
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Antitumor agent-168
Item number: TGM-T89017-10mg
Description: Antitumor agent-168 (compound 21b) disrupts the microtubule networks within tumor cells, leading to G2/M cell cycle arrest and induction of apoptosis. It inhibits the growth of MCF-7 cells with an IC50 value of 1.4 nM. Target: Microtubule Associated
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PPARalpha/gamma agonist 4
Item number: TGM-T89021-10mg
Description: Compound (S)-7, also known as PPARalpha/gamma agonist 4, is a dual potent agonist for PPARalpha and PPARgamma with EC50 values of 0.061 µM and 1.42 µM, respectively. This compound exhibits oral efficacy and operates through an insulin-independent mechanism, featuring mitochondrial pyruvate carrier...
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CK1-IN-4
Item number: TGM-T89036-10mg
Description: CK1-IN-4 (Compound 59) is an inhibitor of casein kinase CK1delta with an IC50 of 2.74 µM. It exhibits neuroprotective activity in SH-SY5Y cells treated with Ethacrynic acid. Target: Casein Kinase
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Dimethylformamide-(S,R,S)-AHPC
Item number: TGM-T89039-10mg
Description: SMARCA2/4-ligand-Linker Conjugate-7 is an E3 ubiquitin ligase ligand-linker conjugate. Target: E3 Ligase Ligand-Linker Conjugate
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Apoptosis inducer 20
Item number: TGM-T89047-10mg
Description: Apoptosisinducer 20 (12) induces cell apoptosis by causing G2/M cell cycle arrest and activating caspase-3/7 during the M-block phase. This compound is a novel indole sulfonamide with anti-proliferative effects against various cancer cells and shows promise for research into new antimitotic drugs....
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RO-76
Item number: TGM-T89060-10mg
Description: RO-76 is a selective partial agonist for the mu opioid receptor (muopioid receptor(µOR)). It binds to the µOR-G-protein complex with an EC50 value of 454 nM. RO-76 reduces the recruitment of beta-Arrestin-1/2 and exhibits analgesic properties. Target: Opioid Receptor
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H2S probe 1
Item number: TGM-T89070-10mg
Description: H2S probe 1 (compound 1NND), a derivative of nitrobenzofurazan (NBD), exhibits antitumor activity. It demonstrates cytotoxicity towards human pancreatic cancer cells, MIA PaCa-2, with an IC50 value of 77.9 nM, and shows high affinity for the human telomeric G-quadruplex with a Kd of 1.72 µM. H2S probe 1...
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