Products from TargetMol
TargetMol, based in Boston, Massachusetts, was founded in 2015 and is a drug screening expert in the life science community. The company offers diverse compound libraries, including FDA-approved libraries, and covers a broad spectrum of small molecule compounds such as inhibitors and agonists as well as recombinant proteins and natural products. TargetMol's products are used by researchers worldwide in areas such as cancer research, neurobiology, inflammation, immunology and metabolism.
More information at: www.targetmol.com
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Somatostatin 1-28
Item number: TGM-TP2124-500ug
Description: Somatostatin receptor agonist, derived from the post-translational cleavage of prosomatostatin. References: Panetta et al (1994) Molecular cloning, functional characterization and chromosomal localization of a human somatostatin receptor (somatostatin receptor type 5) with preferential affinity for...
| MW: | 3149 D |
1,355.00€
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R 892
Item number: TGM-TP2126-1mg
Description: Potent and selective bradykinin B1 receptor antagonist (ID50 values are 2.8 and > 600 nM at B1 and B2 receptors respectively). Exhibits no intrinsic agonist activity and is resistant to aminopeptidase and kininase II (ACE) cleavage. Displays hypertensive activity in vivo. References: Gobeil et al (1996)...
| CAS | 229030-05-1 |
| MW: | 1154.37 D |
170.00€
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RI-STAD 2
Item number: TGM-TP2129-10mg
Description: AKAP disruptor. Selectively binds PKA-RI with high affinity (KD values are 6.2 and 12.1 nM for the RIalpha and beta subunits, respectively) and blocks its interaction with AKAP. Inhibits type I PKA-mediated phosphorylation in live cells. Cell permeable. References: Wang et al (2015) PKA-type I selective...
| MW: | 2401.75 D |
1,646.00€
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26RFa
Item number: TGM-TP2132-1mg
Description: Hypothalamic RFamide-related neuropeptide. Acts as a natural ligand of the orphan receptor GPR103. Exhibits orexigenic acitivity in mice upon central administration. References: Kampe et al (2006) Effect of central administration of QRFP(26) peptide on energy balance and characterization of a second...
| CAS | 881640-56-8 |
| MW: | 2818.18 D |
208.00€
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G3-C12 TFA (848301-94-0 free base)
Item number: TGM-TP1294-10mg
Description: G3-C12 TFA Salt is a specific galectin-3 binding peptide with Ksubdsub of 88 nM and shows anticancer activity. References: Kopansky E, et al. Peptide-directed HPMA copolymer-doxorubicin conjugates as targeted therapeutics for colorectal cancer. J Drug Target. 2011 Dec,19(10):933-43.
| Keywords: | G3-C12 TFA |
| MW: | 1873 D |
From 46.00€
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Foxy-5 TFA(881188-51-8 free base)
Item number: TGM-TP1296-1mg
Description: Foxy-5 is a peptide that mimics the WNT5A protein and is expected to reduce the mobility of the cancer cells. Foxy-5 triggers cytosolic free calcium signaling without affecting beta-catenin activation and it impairs the migration and invasion of epithelial cancer cells[1][2][3]. References: Canesin G,...
| Keywords: | Foxy-5 (TFA) |
| MW: | 808.8 D |
From 93.00€
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Somatostatin acetate
Item number: TGM-TP1302L-100mg
Description: Somatostatin acetate is an endogenously secreted inhibitor of cell proliferation with potential antitumor activity for the study of cancer and neurological disorders. Target: Somatostatin. References: Anthony LB,et al. Opportunities to Improve Symptom Control with Somatostatin Congeners in GEP-NETs: A...
| Keywords: | Somatostatin acetate(51110-01-1 Free base) |
From 51.00€
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RGD peptide (GRGDNP) (TFA) (114681-65-1 free base)
Item number: TGM-TP1311-1mg
Description: RGD peptide (GRGDNP) (TFA) promote apoptosis through activation of conformation changes that enhance pro-caspase-3 activation and autoprocessing. References: Ruoslahti, E., and Öbrink, B. Common principles in cell adhesion Experimental Cell Research 227, 1-11 (1996).
| Keywords: | RGD peptide (GRGDNP) (TFA) |
| MW: | 728.63 D |
From 46.00€
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Cecropin B acetate
Item number: TGM-TP1313L-100mg
Description: Cecropin B acetate induces NF-kappaB activation and suppresses CYP3A29 by disrupting the association of the PXR/retinoid X receptor alpha (RXR-alpha) complex with DNA sequences. Cecropin B acetate exhibits strong antimicrobial activity. Target: Parasite, Retinoid Receptor, P450. References: Zhou X et...
| Keywords: | Cecropin B acetate(80451-05-4 Free base) |
From 82.00€
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AMARA peptide TFA (163560-19-8 free base)
Item number: TGM-TP1314-10mg
Description: AMARA peptide (TFA) is a substrate for salt-induced kinase (SIK) and adenosine activated protein kinase (AMPK). References: Shan T, et al. Lkb1 controls brown adipose tissue growth and thermogenesis by regulating the intracellular localization of CRTC3. Nat Commun. 2016 Jul 27,7:12205.
| Keywords: | AMARA peptide TFA |
| MW: | 1640.84 D |
From 59.00€
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GLP-1 moiety from Dulaglutide
Item number: TGM-TP1316-1mg
Description: The GLP-1 moiety from Dulaglutide is a 31-amino acid fragment of Dulaglutide, a glucagon-like peptide 1 receptor (GLP-1) agonist. References: Anthony Celeste, et al. Anti-pcsk9-glp-1 fusions and methods for use. US 20160369010 A1.
| MW: | 3314.62 D |
From 326.00€
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Galanin (1-16), mouse, porcine, rat TFA
Item number: TGM-TP1317-1mg
Description: Galanin (1-16), mouse, porcine, rat is a potent agonist of the hippocampal galanin receptor with a Kd of 3 nM, and it exhibits high biological activity on locus coeruleus neurons. References: Fisone G, et al. N-terminal galanin-(1-16) fragment is an agonist at the hippocampal galanin receptor. Proc Natl...
| MW: | 1783.9 D |
From 139.00€
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