Products from TargetMol
TargetMol, based in Boston, Massachusetts, was founded in 2015 and is a drug screening expert in the life science community. The company offers diverse compound libraries, including FDA-approved libraries, and covers a broad spectrum of small molecule compounds such as inhibitors and agonists as well as recombinant proteins and natural products. TargetMol's products are used by researchers worldwide in areas such as cancer research, neurobiology, inflammation, immunology and metabolism.
More information at: www.targetmol.com
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CXCR2 antagonist 7
Item number: TGM-T61236-100mg
Description: CXCR2 antagonist 7 (compound 19) is a potent CXCR2 antagonist with strong binding affinity (IC50 = 0.044 µM) and calcium mobilization (IC50 = 0.66 µM) [1]. Target: Others
| MW: | 352.36 D |
From 1,440.00€
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HDAC-IN-32
Item number: TGM-T61248-100mg
Description: HDAC-IN-32 is a highly effective HDAC inhibitor presenting IC50 values of 5.2, 11, and 28 nM for HDAC1, HDAC2, and HDAC6, respectively. This compound demonstrates notable anti-proliferative properties against tumor cells, as well as significant in vivo antitumor efficacy, which can elicit antitumor...
| MW: | 353.41 D |
From 1,440.00€
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Antitubercular agent-16
Item number: TGM-T61252-100mg
Description: Antitubercular agent-16 (Compound 5q) is a potent antitubercular agent exhibiting high efficacy against various strains of M. tuberculosis, including H37Rv, CF16, CF61, CF76, CF152, and CF161, with MIC 90 values ranging from 0.40 to 23.51 µg/mL. Notably, Antitubercular agent-16 demonstrates minimal...
| MW: | 353.52 D |
From 1,440.00€
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Antifungal agent 19
Item number: TGM-T61257-100mg
Description: Antifungal agent 19 demonstrates potent antifungal activity (EC50 = 0.72 µM). Target: Others
| MW: | 354.34 D |
From 1,440.00€
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hCA IX-IN-1
Item number: TGM-T61263-100mg
Description: hCA IX-IN-1 (Compound 6f) is a human carbonic anhydrase ( hCA ) inhibitor with K i values of 331.4, 28.4, 9.4 and 17.8 nM against hCA I, hCA II, hCA IX and hCA XII, respectively. hCA IX-IN-1 shows anticancer activity [1]. Target: Others
| MW: | 354.42 D |
From 1,440.00€
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EGFR/HER2-IN-7
Item number: TGM-T61272-100mg
Description: EGFR/HER2-IN-7 is a highly selective and potent anticancer compound designed to target MCF-7 breast cancer cells by functioning as a dual inhibitor of EGFR/HER2 kinases and DHFR (dihydrofolate reductase), with IC50 values of 0.18 µM for EGFR, 0.146 µM for HER2, and 0.907 µM for DHFR [1]. Target: Others
| MW: | 355.45 D |
From 1,440.00€
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TS010
Item number: TGM-T61279-100mg
Description: TS010 is a highly potent inhibitor of GLO-I, with an IC50 value of 0.57 µM. It holds significant promise for advancements in cancer research [1]. Target: Others
| MW: | 356.36 D |
From 1,440.00€
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CYP121A1-IN-1
Item number: TGM-T61287-100mg
Description: CYP121A1-IN-1 is a potent inhibitor of CYP121A1, demonstrating favorable activity against Mycobacterium tuberculosis (H37Rv MIC 90 ~6.25 µM, ~2.2 µg/mL). It significantly reduces mycocyclosin production by blocking the CYP121A1-mediated conversion of cyclo(l-tyrosyl-l-tyrosyl) to mycocyclosin [1]....
| MW: | 356.42 D |
From 1,440.00€
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CAII-IN-1
Item number: TGM-T61292-100mg
Description: CAII-IN-1 (compound 3n) is a thiosemicarbazide derivative that acts as a potent and selective inhibitor of carbonic anhydrase-II (CA-II), with an IC50 value of 10.3 µM for bovine CA-II. This compound (CAII-IN-1) is useful in research on carbonic anhydrase-associated biological disorders [1]. Target: Others
| MW: | 356.46 D |
From 1,440.00€
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PDE4-IN-5
Item number: TGM-T61295-100mg
Description: PDE4-IN-5 (compound 33a) is a highly potent and selective PDE4 inhibitor with an IC50 value of 3.1 nM, exhibiting excellent skin permeability and a well-characterized binding mechanism. It also shows a notable anti-psoriasis effect [1]. Target: Others
| MW: | 356.46 D |
From 1,440.00€
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LasR-IN-3
Item number: TGM-T61305-100mg
Description: LasR-IN-3, a chemical compound, acts as an inhibitor of LasR in Pseudomonas aeruginosa. It induces structural instability in LasR and causes complete dissociation of its functioning dimeric form [1]. Target: Others
| MW: | 357.41 D |
From 1,440.00€
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Antifungal agent 27
Item number: TGM-T61308-100mg
Description: Antifungal agent 27 (compound 7) is a chemical compound with antifungal properties, exhibiting moderate antibacterial activity and weak antifungal activity against MRSA and C. albicans SS5314, with minimal inhibitory concentration (MIC) values of 8 and 32 µg/mL, respectively [1]. Target: Others
| MW: | 357.47 D |
From 1,440.00€
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