Products from TargetMol
TargetMol, based in Boston, Massachusetts, was founded in 2015 and is a drug screening expert in the life science community. The company offers diverse compound libraries, including FDA-approved libraries, and covers a broad spectrum of small molecule compounds such as inhibitors and agonists as well as recombinant proteins and natural products. TargetMol's products are used by researchers worldwide in areas such as cancer research, neurobiology, inflammation, immunology and metabolism.
More information at: www.targetmol.com
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PLP_Snyder530
Item number: TGM-T61500-100mg
Description: PLP_Snyder530 is a potent papain-like protease (PL pro) inhibitor that induces conformational changes in SARS-CoV-2 papain-like protease, thereby inhibiting SARS-CoV-2 replication, it can be used for SARS-CoV-2 research [1]. Target: Others
| MW: | 372.46 D |
From 1,440.00€
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alpha-Glucosidase-IN-15
Item number: TGM-T61503-100mg
Description: alpha-Glucosidase-IN-15 (Compound 14B) exhibits potent alpha-glucosidase inhibitory activity with an IC50 value of 3.34 µM and possesses antidiabetic properties [1]. Target: Others
| MW: | 372.53 D |
From 1,440.00€
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NBI-31772 hydrate
Item number: TGM-T61506-100mg
Description: NBI-31772 hydrate is a powerful inhibitor of the interaction between insulin-like growth factor (IGF) and IGF-binding proteins (IGFBPs). It acts as a nonpeptide ligand, effectively releasing bioactive IGF-I from the IGF-I/IGFBP-3 complex (Ki values for all six human subtypes range from 1-24 nM). This...
| MW: | 372.82 D |
From 1,080.00€
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PIM-1/HDAC-IN-1
Item number: TGM-T61510-100mg
Description: PIM-1/HDAC-IN-1 (compound 4d) is a potent PIM-1 inhibitor with an IC50 of 343.87 nM, and it exhibits strong inhibitory activity and selectivity against HDAC 1 and HDAC 6, with IC50 values of 63.65 and 62.39 nM, respectively. Additionally, it induces apoptosis and causes G2/M phase cell cycle arrest in...
| MW: | 373.4 D |
From 1,440.00€
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FT3967385
Item number: TGM-T61512-100mg
Description: FT3967385 is a newly developed compound that functions as a USP30 inhibitor, emulating the genetic deficiency of USP30. This inhibition serves as a catalyst for the amplification of mitochondrial ubiquitylation through the PINK1-PARKIN pathway. Target: Others
| MW: | 373.41 D |
From 1,440.00€
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Enpp-1-IN-12
Item number: TGM-T61514-100mg
Description: Enpp-1-IN-12 (compound 43), an orally active and potent inhibitor of ecto-nucleotide pyrophosphatase/phosphodiesterase 1 (ENPP1) with a K_i of 41 nM, exhibits anti-tumor activity [1]. Target: Others
| MW: | 373.43 D |
From 1,440.00€
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alpha-Glucosidase-IN-18
Item number: TGM-T61519-100mg
Description: alpha-Glucosidase-IN-18 (7B) is an orally active alpha-glucosidase inhibitor with an IC50 value of 3.96 µM, exhibiting antidiabetic properties [1]. Target: Others
| MW: | 373.47 D |
From 1,440.00€
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Nrf2/HO-1 activator 2
Item number: TGM-T61522-100mg
Description: Nrf2/HO-1 activator 2 (compound 13m), a difluoro-substituted derivative, is a highly potent activator of Nrf2/HO-1 with substantial neuroprotective and antioxidant properties. It functions by activating the Nrf2/HO-1 pathway through the phosphorylation of ERK1/2, JNK, or Akt in PC12 cells and is useful...
| MW: | 374.33 D |
From 1,440.00€
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CK2 inhibitor 3
Item number: TGM-T61629-100mg
Description: CK2 inhibitor 3 is a highly potent inhibitor of protein kinase CK2, exhibiting an IC50 value of 280 nM. It effectively inhibits the intracellular activity of CK2 and displays a notable impact on the viability of tumor cells. Moreover, CK2 inhibitor 3 demonstrates exceptional selectivity among a diverse...
| MW: | 381.2 D |
From 1,440.00€
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Glucosylceramide synthase-IN-3
Item number: TGM-T61632-100mg
Description: Glucosylceramide synthase-IN-3 (compound BZ1) is a highly potent, brain-penetrant, and orally active inhibitor of glucosylceramide synthase (GCS), with an IC50 value of 16 nM for human GCS, and has potential applications in Gaucher's disease research [1] [2]. Target: Others
| MW: | 381.4 D |
From 1,440.00€
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Antibacterial agent 77
Item number: TGM-T61640-100mg
Description: Antibacterial agent 77 (compound 12) is an antibacterial agent [1]. Target: Others
| MW: | 381.53 D |
From 1,440.00€
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Utrophin modulator 1
Item number: TGM-T61645-100mg
Description: Utrophin Modulator 1 (UM1) is a highly effective agent that upregulates utrophin protein levels, displaying an EC 50 of 0.11 µM. Its application in the investigation of Duchenne Muscular Dystrophy (DMD) has been well-established [1]. Target: Others
| MW: | 382.42 D |
From 1,440.00€
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