78 products were found matching "K05181"!

Alphenal (Cay-26918) is an analytical reference standard categorized as a barbiturate. This product is intended for research and forensic applications.Formal Name: 5-phenyl-5-(2-propen-1-yl)-2,4,6(1H,3H,5H)-pyrimidinetrione. CAS Number: 115-43-5. Molecular Formula: C13H12N2O3. Formula Weight: 244.2. Purity: >95%....

Chrodrimanin B is a meroterpenoid fungal metabolite that has been found in Talaromyces species. It has insecticidal activity against third instar silkworm larvae (LD50 = 10 µg/g of diet). Chrodrimanin B selectively inhibits the silkworm GABA receptor RDL (IC50 = 1.13 nM) over human alpha1beta2gamma2...

Clobazam (Cay-14262) is an analytical reference standard categorized as a benzodiazepine. Clobazam is regulated as a Schedule IV compound in the United States. This product is intended for research and forensic applications.Formal Name: 7-chloro-1-methyl-5-phenyl-1H-1,5-benzodiazepine-2,4(3H,5H)-dione. CAS Number:...

Bretazenil (Cay-37274) is an analytical reference standard categorized as a GABAA receptor positive allosteric modulator. Bretazenil has anxiolytic-like effects in mice. It induces self-administration in rhesus monkeys but has a lower physical dependence liability in mice compared with benzodiazepines. This product...

Adinazolam (Cay-18205) is an analytical reference material categorized as a benzodiazepine. This product is intended for research and forensic applications.Formal Name: 8-chloro-N,N-dimethyl-6-phenyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepine-1-methanamine. CAS Number: 37115-32-5. Molecular Formula: C19H18ClN5....

N-Desmethylclobazam (Cay-18564) is an analytical reference material that is structurally categorized as a benzodiazepine. It is a major active metabolite of clobazam, produced primarily by the action of cytochrome P450 isoform 3A4. N-Desmethylclobazam positively modulates GABAA receptors (EC50s range from 98 to 151...

Cinolazepam (Cay-20529) is an analytical reference material categorized as a benzodiazepine. This product is intended for research and forensic applications.Formal Name: 7-chloro-5-(2-fluorophenyl)-2,3-dihydro-3-hydroxy-2-oxo-1H-1,4-benzodiazepine-1-propanenitrile. CAS Number: 75696-02-5. Molecular Formula:...

Tofisopam (Cay-22026) is an analytical reference standard categorized as a benzodiazepine. This product is intended for research and forensic applications.Formal Name: 1-(3,4-dimethoxyphenyl)-5-ethyl-7,8-dimethoxy-4-methyl-5H-2,3-benzodiazepine. CAS Number: 22345-47-7. Molecular Formula: C22H26N2O4. Formula Weight:...

Desmethylclotiazepam (Cay-27838) is an analytical reference standard categorized as a thienodiazepine. It is an active metabolite of clotiazepam. This product is intended for research and forensic applications.Formal Name: 5-(2-chlorophenyl)-7-ethyl-1,3-dihydro-2H-thieno[2,3-e]-1,4-diazepin-2-one. CAS Number:...

Milbemectin is a mixture of milbemycin A3 (30%, Cay-18360) and milbemycin A4 (70%, Cay-17155) that has acaricidal and nematocidal activity against adult spider mites, spider mite eggs, and C. elegans with IC50 values of 5.3, 41.1, and 9.5 µg/ml, respectively. It acts as an allosteric agonist of the Drosophila RDL...

Anti-GABA(A) Receptor beta 3 pS408/pS409 Antibody is directed against rat GABA(A) Receptor beta 3. The antibody was affinity purified from monospecific antiserum by immunoaffintiy purification. Immunolabeling of the GABAA band is completely blocked by the phospho-peptide used as antigen but not by the corresponding...

Bretazenil is a positive allosteric modulator of GABAA receptors with anticonvulsant and anxiolytic activity. It potentiates GABA-gated chloride currents in rat cortical neurons and in HEK293 cells expressing alpha1beta1gamma2 subunit-containing GABAA receptors (EC50s = 60 and 10 nM, respectively). Bretazenil...