93 products were found matching "K04280"!

Recombinant CHO-K1 cells stably overexpress human gonadotropin releasing hormone receptor (GNRHR) on the surface and contain high levels of G protein Galphaq to couple with the receptor in downstream signaling pathways.

A GnRH receptor antagonist (Kis = 6, 2.2, and 3.8 nM for the human, mouse, and rat receptors, respectively), selective for the GnRH receptor over a panel of 43 receptors, ion channels, and enzymes at 1 µM, prevents GnRH-induced increases in inositol phosphate production in HEK293 cells expressing the human GnRH...

Fertirelin is a peptide agonist of the gonadotropin-releasing hormone receptor (GnRHR) and a derivative of GnRH. It binds to GnRHR in CHO cells expressing the human receptor (Ki = 0. nM). In vivo, fertirelin (200 µg/animal) increases serum levels of luteinizing hormone and induces luteinization of follicular cysts...

Leuprorelin is a synthetic gonadotropin-releasing hormone (GnRH) receptor agonist. It is a long-acting agent that, after an initial increase in sex hormone levels, decreases the level of circulating gonadotropins and sex hormones. Formulations containing leuprorelin have been used in the treatment of...

Cetrorelix is a synthetic peptide antagonist of the gonadotropin-releasing hormone receptor (GnRHR) with a Kd value of 0.2 nM for radioligand binding to murine LTK- cells expressing human GnRHR. It inhibits the activation of hGnRHR and a downstream luciferase reporter gene in murine LTK- cells by the GnRHR agonist...

Description: Nafarelin acetate(76932-56-4 free base) (RS-94991-298) is a GnRH agonist that acts as an analog of GnRH. Nafarelin acetate(76932-56-4 free base) causes a decrease in the pituitary secretion of gonadotropins luteinizing hormone (LH) and follicle-stimulating hormone (FSH). It may be used in the treatment...

Protein function: Receptor for gonadotropin releasing hormone (GnRH) that mediates the action of GnRH to stimulate the secretion of the gonadotropic hormones luteinizing hormone (LH) and follicle- stimulating hormone (FSH). This receptor mediates its action by association with G-proteins that activate a...

Protein function: Receptor for gonadotropin releasing hormone (GnRH) that mediates the action of GnRH to stimulate the secretion of the gonadotropic hormones luteinizing hormone (LH) and follicle- stimulating hormone (FSH). This receptor mediates its action by association with G-proteins that activate a...

Cetrorelix is a gonadotropin-releasing hormone (GnRH) analog that inhibits LHRH and GnRH. Cetrorelix exhibits anti-inflammatory activity and has been used clinically as a treatment for infertility due to its suppression of FSH and LH levels. In animal models of benign prostatic hyperplasia (BPH), cetrorelix...

0.5 mg/ml in 1X TBS, pH7.3, with 0.5% BSA (US sourced) and 0.02% sodium azide. Additional name(s) for this target protein: Gonadotropin-releasing hormone receptor, GRHR, LRHR Protein function: Receptor for gonadotropin releasing hormone (GnRH) that mediates the action of GnRH to stimulate the secretion of the...