368 products were found matching "K04277"!
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Human Cannabinoid receptor 1 Protein-VLP
Item number: KT-CNR-HM001-100UG
Recombinant Human Cannabinoid receptor 1 Protein-VLP is expressed from HEK293.It contains Met1-Leu472. The CB1 receptor also plays an important role in the gut-brain axis control of appetite and satiety. The combined effect of peripheral CB1 activation is to promote appetite, energy storage, and energy preservation...
| Keywords: | CB-R,CB R,CBR,CB1,CANN6,CANN6CB1R,Cannabinoid R1,CB1K5,CB1R,CB-RCB1cannabinoid receptor 1,central cannabinoid... |
| Expressed in: | Human cells |
| Origin: | human |
| MW: | 52.9 kD |
2,295.00€
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N-Arachidonoyl Dopamine
Item number: Cay90057-5
N-Arachidonoyl dopamine (NADA) is an arachidonoyl amino acid and cannabinoid (CB) receptor 1 agonist (Ki = 250 nM in rat brain membranes, which highly express CB1 receptors). It is selective for CB1 over CB2 receptors (Ki = 12,000 nM in rat spleen membranes, which highly express CB2 receptors). NADA induces...
| Keywords: | NADA, N-[2-(3,4-dihydroxyphenyl)ethyl]-5Z,8Z,11Z,14Z-eicosatetraenamide |
| Application: | CB1 agonist |
| CAS | 199875-69-9 |
| MW: | 439.6 D |
From 74.00€
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ADB-5'F-BUTINACA
Item number: Cay37761-1
ADB-5'F-BUTINACA (Cay-37761) is an analytical reference standard categorized as a synthetic cannabinoid. This product is intended for research and forensic applications.Formal Name: (S)-N-(1-amino-3,3-dimethyl-1-oxobutan-2-yl)-1-butyl-5-fluoro-1H-indazole-3-carboxamide. Molecular Formula: C18H25FN4O2. Formula...
| Keywords: | ADB-B-5'F-INACA, ADB-BUT-5'F-INACA, (S)-N-(1-amino-3,3-dimethyl-1-oxobutan-2-yl)-1-butyl-5-fluoro-1H-indazole-3-carboxamide |
| Application: | Analytical reference standard, synthetic cannabinoid |
| MW: | 348.4 D |
From 111.00€
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AM251
Item number: Cay71670-10
AM251 is a cannabinoid 1 (CB1) receptor 1 antagonist. It binds to CB1 receptors in rat forebrain membrane preparations (Ki = 7.5 nM) and is selective over CB2 receptors in mouse spleen preparations (Ki = 2,290 nM) in radioligand binding assays. AM251 inhibits GTPgammaS binding induced by the CB receptor agonist CP...
| Keywords: | 1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-1-piperidinyl-1H-pyrazole-3-carboxamide |
| Application: | SR 141716A analog |
| CAS | 183232-66-8 |
| MW: | 555.2 D |
From 67.00€
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JWH 116
Item number: Cay13977-1
JWH 116 (Cay-13977) is a synthetic cannabinoid (CB) receptor ligand from the naphthoylindole family. It is the indole 2-ethyl derivative of the related compound JWH 018 (Cay-10900 and 13169) and has a Ki value of 52 nM for the CB1 receptor. This product is intended for research and forensic applications.Formal Name:...
| Keywords: | (2-ethyl-1-pentyl-1H-indol-3-yl)-1-naphthalenyl-methanone |
| Application: | Analytical reference standard, synthetic cannabinoid, CB1 receptor agonist |
| CAS | 619294-64-3 |
| MW: | 369.5 D |
From 61.00€
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CB-25
Item number: TGM-T78083-2mg
Description: CB-25 is a partial agonist ligand of CB1 cannabinoid receptors, augmenting Forskolin-induced cAMP formation in cancer cells, though not affecting hCB1-CHO cells [1]. Target: Cannabinoid Receptor. Smiles: O=C(NC1CC1)CCCCCCCCCC OC2=CC(O)=CC(=C2)CCCCC
| Application: | CB1 receptor inverse agonist |
| CAS | 869376-63-6 |
| MW: | 403.6 D |
97.00€
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JWH 080
Item number: TGM-T84720-10mg
Description: JWH 080 is a synthetic cannabinoid that exhibits affinity for both central CB1 receptors (Ki = 5.6 nM) and peripheral CB2 receptors (Ki = 2.2 nM) in vitro. The in vivo physiological and toxicological characteristics of this compound remain uncharacterized. It is designed for forensic and research...
| Application: | Synthetic cannabinoid |
| CAS | 210179-44-5 |
| MW: | 357.4 D |
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PSB-SB1202
Item number: TGM-T84440-10mg
Description: PSB-SB1202 (Compound 21a), a phenyl coumarin compound, acts as a CB1/CB2 agonist. It demonstrates EC50 values of 56 and 14 nM and K i values of 32 and 49 nM for CB1 and CB2 receptors, respectively [1]. Target: Others. Smiles: O(C)C1=C2C(=CC(CCCCC)=C1)OC(=O)C(CC3=C(OC)C=CC=C3)=C2
| Application: | CB1 / CB2 receptor agonist |
| CAS | 1399049-60-5 |
| MW: | 366.45 D |
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JWH 387
Item number: TGM-T84462-10mg
Description: JWH 387, a potent analgesic cannabimimetic belonging to the naphthoylindole family, serves as a strong cannabinoid (CB) agonist targeting both central CB1 and peripheral CB2 receptors with Ki values of 1.2 and 1.1 nM, respectively. This compound is designed for research and forensic applications....
| Application: | analgesic cannabimimetic, non-selective potent cannabinoid agonist |
| CAS | 1366067-59-5 |
| MW: | 420.3 D |
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JWH 176
Item number: TGM-T84463-10mg
Description: JWH-176 is a cannabimimetic indene hydrocarbon, exhibiting high affinity for the central cannabinoid (CB1) receptor (Ki= 26 nM), originally synthesized to investigate hydrogen bonding and aromatic stacking's roles in CB1 receptor docking studies. Intended for forensic and research applications, this...
| Application: | Cannabimimetic indene hydrocarbon (high CB1 receptor affinity) |
| CAS | 619294-62-1 |
| MW: | 324.5 D |
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Cannabipiperidiethanone
Item number: TGM-T84468-10mg
Description: Cannabipiperidiethanone, a synthetic cannabinoid structurally similar to JWH 250 and AM2233, has been detected in prohibited "herbal" blends in Japan. It exhibits affinity for CB1 and CB2 receptors with IC50 values of 591 nM and 968 nM, respectively. Compared to JWH 250, its affinities for CB1 and CB2...
| Application: | Synthetic cannabinoid (CB1 / CB2 binding) |
| CAS | 1345970-43-5 |
| MW: | 376.5 D |
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CB-52
Item number: TGM-T84515-10mg
Description: CB-52 acts as a neutral antagonist and ligand for the CB2 cannabinoid receptor [1]. Target: Others. Smiles: O(CCCCCCCCCCC(NC1CC1)=O)C2=C(CCCCCC)C=CC(O)=C2
| Application: | CB1 receptor partial agonist, CB2 receptor neutral antagonist |
| CAS | 869376-90-9 |
| MW: | 417.62 D |
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