- Search results for K04265
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63 products were found matching "K04265"!
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Item number: CSB-CF001375HU.100
Organism: Homo sapiens (Human). Source: in vitro E.coli expression system. Expression Region: 1-326aa. Protein Length: Full Length. Tag Info: N-terminal 10xHis-tagged. Target Protein Sequence: MPPSISAFQA AYIGIEVLIA LVSVPGNVLV IWAVKVNQAL RDATFCFIVS LAVADVAVGA LVIPLAILIN IGPQTYFHTC LMVACPVLIL TQSSILALLA IAVDRYLRVK...
Keywords: | ADORA1, Adenosine receptor A1, Recombinant Human Adenosine receptor A1 (ADORA1) |
Application: | Activity not tested |
Expressed in: | E.coli in vitro |
Origin: | human |
MW: | 39.3 kD |
From 1,413.00€
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Item number: CSB-RA224168A0HU.100
Isotype: Rabbit IgG. Buffer: Rabbit IgG in phosphate buffered saline, pH 7.4, 150mM NaCl, 0.02% sodium azide and 50% glycerol. Storage: Upon receipt, store at -20°C or -80°C. Avoid repeated freeze. Purification Method: Affinity-chromatography. Target Name: ADORA1. Antigen Species: Human
Keywords: | Anti-ADORA1, Anti-Adenosine receptor A1, Adenosine receptor A1, ADORA1, ADORA1 Recombinant Monoclonal Antibody |
Application: | ELISA, WB, IHC, FC |
Host: | Rabbit |
Species reactivity: | human |
From 201.00€
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Item number: Cay21972-10
DPCPX is an adenosine A1 receptor antagonist (Ki = 0.3 nM). It is selective for the adenosine A1 receptor over the adenosine A2 receptor (Ki = 340 nM). DPCPX (0.03 and 1 µM) increases the force of contractions in isolated guinea pig left auricles and inhibits decreases in contraction forces induced by the adenosine...
Keywords: | 1,3-Dipropyl-8-cyclopentylxanthine, 8-Cyclopentyl-1,3-dipropylxanthine, PD 116948,... |
Application: | Adenosine A1 receptor antagonist |
CAS | 102146-07-6 |
MW: | 304.4 D |
From 40.00€
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Item number: Cay37776-10
MIPS521 is an adenosine A1 receptor positive allosteric modulator. It binds to adenosine A1 receptors (Kb = 11 µM) and enhances adenosine-induced inhibition of forskolin-induced cAMP production in CHO cells expressing recombinant human adenosine A1 receptors when used at concentrations ranging from 0.3 to 30 µM. In...
Keywords: | [2-amino-4-[3,5-bis(trifluoromethyl)phenyl]-3-thienyl](4-chlorophenyl)-methanone |
Application: | Adenosine A1 receptor positive allosteric modulator |
CAS | 1146188-19-3 |
MW: | 449.8 D |
From 90.00€
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Item number: ELK-ELK6925.48
The test principle applied in this kit is Sandwich enzyme immunoassay. The microtiter plate provided in this kit has been pre-coated with an antibody specific to Rat ADORA1. Standards or samples are added to the appropriate microtiter plate wells then with a biotin-conjugated antibody specific to Rat ADORA1. Next,...
Keywords: | Adora1, Adenosine receptor A1 |
Application: | ELISA |
Species reactivity: | rat |
From 365.00€
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Item number: Cay21420-5
5'-N-Ethylcarboxamidoadenosine (NECA) is an adenosine analog that acts as an agonist of adenosine receptors (Kis = 1,880, 6,660, and 3.5 nM for human adenosine subtypes A1, A2A, and A3, respectively). NECA is reported to act as a potent vasodilator and can inhibit platelet aggregation by increasing cAMP (EC50 = 3.1...
Keywords: | Adenosine 5'-ethylcarboxamide, NECA, 1-(6-amino-9H-purin-9-yl)-1-deoxy-N-ethyl-beta-D-ribofuranuronamide, hydrate |
Application: | Adenosine receptor agonist |
MW: | 308.3 D |
From 43.00€
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Item number: Cay15612-10
2-Chloroadenosine (CADO) is a metabolically stable analog of adenosine that binds to adenosine A1, A2A, and A3 receptors with Ki values of 300, 80, and 1,900 nM, respectively. CADO has been used to activate adenosine receptors in the thalamus, generating anticonvulsive activity in a rat model of generalized...
Keywords: | Antibiotic AT-265B, CADO, NSC 36896, 2-chloro-adenosine |
Application: | Adenosine A1/A2A/A3 receptor agonist |
CAS | 146-77-0 |
MW: | 301.7 D |
From 43.00€
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Item number: Cay21745-25
Theobromine is a methylxanthine alkaloid and derivative of caffeine (Cay-14118) that has been found in cocoa beans and has diverse biological activities. It is an adenosine A1 receptor antagonist (IC50s = 200-280 µM in radioligand binding assays using rat brain membranes). Theobromine (150 µg/ml) increases AMPK...
Keywords: | Diurobromine, NSC 5039, SC-15090, 3,7-dihydro-3,7-dimethyl-1H-purine-2,6-dione |
Application: | Adenosine receptor antagonist |
CAS | 83-67-0 |
MW: | 180.2 D |
From 43.00€
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Item number: Cay14118-5
Caffeine is a methylxanthine alkaloid naturally found in various plant parts that acts as an antagonist at central adenosine receptors at relevant physiological concentrations (IC50 = ~30 µM). It alters fatigue, mood, alertness, motor reaction time, vascular hemodynamics, and pain sensation. Caffeine has also been...
Keywords: | Methyltheobromine, NSC 5036, 3,7-dihydro-1,3,7-trimethyl-1H-purine-2,6-dione |
Application: | Adenosine receptor antagonist |
CAS | 58-08-2 |
MW: | 194.2 D |
From 34.00€
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Item number: Cay15593-100
5'-Deoxy-5'-methylthioadenosine (MTA) is an intermediate in the generation of adenine and methionine that is produced by the decarboxylation of S-adenosylmethionine. This nucleoside is a potent agonist of adenosine receptors (Kis = 0.15, 1.13, 13.9, and 0.68 µM for A1, A2A, A2B, and A3, respectively). At higher...
Keywords: | 5'-S-Methylthioadenosine, MTA, NSC 335422, Vitamin L2, 5'-S-methyl-5'-thio-adenosine |
Application: | Intermediate, Adenosine receptor agonist |
CAS | 2457-80-9 |
MW: | 297.3 D |
From 56.00€
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Item number: Cay34348-50
7-Methylxanthine is an adenosine A1 receptor antagonist and active metabolite of theobromine (Cay-21745) and caffeine (Cay-14118). It inhibits binding of the adenosine A1 receptor agonist cyclohexyladenosine in rat cerebral cortical membranes in a concentration-dependent manner. 7-Methylxanthine (300 mg/kg) inhibits...
Keywords: | 7-MX, NSC 7861, 3,7-dihydro-7-methyl-1H-purine-2,6-dione |
Application: | Active theobromine / caffeine metabolite, Adenosine A1 receptor antagonist |
CAS | 552-62-5 |
MW: | 166.1 D |
From 66.00€
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Item number: Cay11940-10
KW 3902 is an antagonist of the adenosine A1 receptor (Ki = 0.19 nM). It displays 890-fold selectivity for A1 receptors over A2A receptors and has no activity at A3 receptors. KW 3902 less potently inhibits human organic anion transporter 1 (OAT1, Ki = 7.82 µM). KW 3902 exhibits renal protective effects during...
Keywords: | MK-7418, Rolofylline, 8-(hexahydro-2,5-methanopentalen-3a(1H)-yl)-3,9-dihydro-1,3-dipropyl-1H-purine-2,6-dione |
Application: | Adenosine A1 receptor antagonist |
CAS | 136199-02-5 |
MW: | 356.5 D |
From 43.00€
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