- Search results for K04238
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30 products were found matching "K04238"!
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Item number: Cay22911-1
Suvorexant (Cay-22911) is an analytical reference standard categorized as a diazepane sedative. Formulations containing suvorexant show abuse potential similar to zolpidem (Cay-15792) in recreational polydrug users with a history of sedative and psychedelic drug use. Suvorexant is regulated as a Schedule IV compound...
Keywords: | MK-4305,... |
Application: | Analytical reference standard, Diazepane sedative, Orexin receptor antagonist |
CAS | 1030377-33-3 |
MW: | 450.9 D |
From 76.00€
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Item number: ARG64584.100
Protein function: Moderately selective excitatory receptor for orexin-A and, with a lower affinity, for orexin-B neuropeptide. Seems to be exclusively coupled to the G(q) subclass of heteromeric G proteins, which activates the phospholipase C mediated signaling cascade. [The UniProt Consortium]
Keywords: | Anti-Ox1R, Anti-Ox1-R, Anti-Ox-1-R, Anti-HCRTR1, Anti-Orexin receptor type 1, Anti-Hypocretin receptor type 1 |
Application: | ELISA, WB |
Host: | Goat |
Species reactivity: | human, mouse, rat |
784.00€
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Item number: G-HUFI00849.96
Application: | ELISA |
Species reactivity: | human |
641.00€
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Item number: NSJ-R35702-100UG
0.5 mg/ml in 1X TBS, pH7.3, with 0.5% BSA (US sourced) and 0.02% sodium azide. Additional name(s) for this target protein: Hypocretin receptor-1, HCRTR1 Protein function: Moderately selective excitatory receptor for orexin-A and, with a lower affinity, for orexin-B neuropeptide. Seems to be exclusively coupled to...
Keywords: | Anti-Ox1R, Anti-Ox1-R, Anti-Ox-1-R, Anti-HCRTR1, Anti-Orexin receptor type 1, Anti-Hypocretin receptor type 1, Orexin... |
Application: | WB, ELISA (peptide) |
Host: | Goat |
Species reactivity: | human |
755.00€
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Item number: NSJ-R36388-100UG
0.5 mg/ml in 1X TBS, pH7.3, with 0.5% BSA (US sourced) and 0.02% sodium azide. Additional name(s) for this target protein: Hypocretin (orexin) receptor 1, HCRTR1 Protein function: Moderately selective excitatory receptor for orexin-A and, with a lower affinity, for orexin-B neuropeptide. Seems to be exclusively...
Keywords: | Anti-Ox1R, Anti-Ox1-R, Anti-Ox-1-R, Anti-HCRTR1, Anti-Orexin receptor type 1, Anti-Hypocretin receptor type 1, Orexin... |
Application: | WB, ELISA (peptide) |
Host: | Goat |
Species reactivity: | human, mouse, rat |
755.00€
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Item number: Cay13638-1
Almorexant is a dual antagonist of orexin 1 receptor (OX1R) and OX2R (Kis = 4.7 and 0.9 nM, respectively, in a radioligand binding assay). It decreases the latency to persistent non-rapid eye movement (NREM) sleep and increases the duration of NREM and REM sleep in male rats when administered at a dose of 100 mg/kg....
Keywords: | ACT 078573,... |
Application: | HCRTR1/2 antagonist |
CAS | 913358-93-7 |
MW: | 549 D |
From 60.00€
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Item number: Cay18495-1
Orexin receptors 1 (OX1R) and OX2R mediate the action of the neuropeptides orexin A and orexin B. TCS 1102 is a dual antagonist of both OX1R and OX2R (Kis = 0.2 and 3 nM, respectively). It is a poor substrate for P-glycoprotein and, as a result, demonstrates good brain penetration when administered...
Keywords: | (2S)-N-[1,1'-biphenyl]-2-yl-1-[2-[(1-methyl-1H-benzimidazol-2-yl)thio]acetyl]-2-pyrrolidinecarboxamide |
Application: | OX1R / OX2R antagonist |
CAS | 916141-36-1 |
MW: | 470.6 D |
From 43.00€
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Item number: E-AB-12828.120
The protein encoded by this gene is a G-protein coupled receptor involved in the regulation of feeding behavior. The encoded protein selectively binds the hypothalamic neuropeptide orexin A. A related gene (HCRTR2) encodes a G-protein coupled receptor that binds orexin A and orexin B. Protein function: Moderately...
Keywords: | Anti-Ox1R, Anti-Ox1-R, Anti-HCRTR1, Anti-Ox-1-R, Anti-Orexin receptor type 1, Anti-Hypocretin receptor type 1, HCRTR1... |
Application: | IHC, ELISA |
Host: | Rabbit |
Species reactivity: | human, mouse, rat |
From 71.00€
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Item number: E-AB-16019.120
The protein encoded by this gene is a G-protein coupled receptor involved in the regulation of feeding behavior. The encoded protein selectively binds the hypothalamic neuropeptide orexin A. A related gene (HCRTR2) encodes a G-protein coupled receptor that binds orexin A and orexin B. Protein function: Moderately...
Keywords: | Anti-Ox1R, Anti-Ox1-R, Anti-HCRTR1, Anti-Ox-1-R, Anti-Orexin receptor type 1, Anti-Hypocretin receptor type 1, HCRTR1... |
Application: | IHC, ELISA |
Host: | Rabbit |
Species reactivity: | human, mouse, rat |
From 71.00€
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Item number: Cay19145-1
SB-334867 is an antagonist of the orexin 1 receptor (OX1R, KB = 39.8 nM) that is selective for OX1R over OX2R (KB = 1,995.3 nM). It reduces food intake and increases resting duration in rats, as well as inhibits orexin-A-induced increases in food intake, when administered at a dose of 30 mg/kg. SB-334867 (10 mg/kg)...
Keywords: | N-(2-methyl-6-benzoxazolyl)-N'-1,5-naphthyridin-4-yl-urea |
Application: | OX1 receptor antagonist |
CAS | 792173-99-0 |
MW: | 319.3 D |
From 34.00€
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Item number: Cay21270-1
SB-674042 is a potent and selective non-peptide orexin 1 receptor (OX1R) antagonist (Kd = 5.03 and 3.76 nM in whole cell binding and membrane-based assays, respectively). In calcium mobilization studies, it was >100-fold selective for OX1 over OX2 and did not show significant affinity for serotonergic, dopaminergic,...
Keywords: | [5-(2-fluorophenyl)-2-methyl-4-thiazolyl][(2S)-2-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1-pyrrolidinyl]-methanone |
Application: | OX1 receptor antagonist |
CAS | 483313-22-0 |
MW: | 448.5 D |
From 46.00€
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Item number: Cay22961-10
SB-408124 is a potent antagonist of orexin 1 receptors (OX1Rs) with a Ki value of 26.9 nM in a calcium mobilization assay using CHO cells that stably express human OX1R. It is selective for OX1R over OX2R, with Kd values of 21.7 and 1,704 nM, respectively, in a radioligand binding assay. In vivo co-perfusion of...
Keywords: | N-(6,8-difluoro-2-methyl-4-quinolinyl)-N'-[4-(dimethylamino)phenyl]-urea |
Application: | OX1R antagonist |
CAS | 288150-92-5 |
MW: | 356.4 D |
From 109.00€
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