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CDN1163
CDN1163

Item number: Cay31123-1

CDN1163 is an allosteric activator of sarcoplasmic/endoplasmic reticulum Ca2+-ATPase 2 (SERCA2) that enhances calcium uptake in endoplasmic reticulum (ER) vesicles when used at concentrations ranging from 1 to 10 µM. It decreases peroxide-induced cell death in HEK293 cells. CDN1163 (50 mg/kg) increases calcium...
Keywords: 4-(1-methylethoxy)-N-(2-methyl-8-quinolinyl)-benzamide
Application: Allosteric SERCA2 activator
CAS 892711-75-0
MW: 320.4 D
From 49.00€ *
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CDN1163
CDN1163

Item number: TGM-T7373-100mg

Description: CDN1163 is a small molecule activator of sarco/endoplasmic reticulum Ca2+-ATPase (SERCA). Target: Calcium Channel. Smiles: CC(C)Oc1ccc(cc1)C(=O)Nc1cccc2ccc(C)nc12. References: Rizwan, Qaisar, Shylesh, et al. Restoration of SERCA ATPase prevents oxidative stress-related muscle atrophy and weakness.[J]....
Application: Allosteric SERCA2 activator
CAS 892711-75-0
MW: 320.39 D
From 35.00€ *
Review