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LUF6000
LUF6000

Item number: TGM-T15791-100mg

Description: LUF6000 is an allosteric modulator of the human A3 adenosine receptor (AR). Target: Others. Smiles: Clc1ccc(Nc2nc3ccccc3c3nc([nH]c23)C2CCCCC2)cc1Cl. References: Gao ZG, Verzijl D, Zweemer A et al. Functionally biased modulation of A(3) adenosine receptor agonist efficacy and potency by...
Application: Adenosine receptor A3 agonist
CAS 890087-21-5
MW: 411.33 D
From 325.00€ *
Review
LUF6000
LUF6000

Item number: Cay28437-1

LUF6000 is a positive allosteric modulator of adenosine A3 receptors. It reduces dissociation of the agonist I-AB-MECA from A3 receptors and increases the efficacy, but not potency, of 2-Cl-IB-MECA-induced inhibition of forskolin-stimulated cAMP accumulation by 45% in CHO cells expressing the human receptor when...
Keywords: 2-cyclohexyl-N-(3,4-dichlorophenyl)-3H-imidazo[4,5-c]quinolin-4-amine
Application: Adenosine receptor A3 agonist
CAS 890087-21-5
MW: 411.3 D
From 111.00€ *
Review