4 products were found matching "868540-17-4"!
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Carfilzomib
Item number: Cay17554-5
Carfilzomib is a second-generation, irreversible, peptide epoxyketone class proteasome inhibitor that targets the chymotrypsin-like beta5 subunit of the constitutive 20S proteasome (IC50 = 5.2 nM) and the beta5i subunit of the immunoproteasome 20Si (LMP7, IC50 = 14 nM) with minimal cross reactivity to other...
| Keywords: | PR-171,... |
| Application: | Proteasome PSMB5 inhibitor |
| CAS | 868540-17-4 |
| MW: | 719.9 D |
From 43.00€
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Carfilzomib
Item number: LKT-C0271.1
Carfilzomib, a tetrapeptide epoxyketone, is an epoxomicin derivate with potential antineoplastic activity. Carfilzomib irreversibly binds to and inhibits the chymotrypsin-like activity of the 20S proteasome, an enzyme responsible for degrading a large variety of cellular proteins.
| Keywords: | PR-171,... |
| Application: | Proteasome chymotrypsin-like activity inhibitor |
| CAS | 868540-17-4 |
| MW: | 719.91 D |
From 139.00€
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![Carfilzomib [PR-171]](https://www.biomol.com/media/image/71/4c/e3/AG-CR1-3669-M001_200x200.png "Carfilzomib [PR-171]")
Carfilzomib [PR-171]
Item number: AG-CR1-3669-M005
Synthetic. Chemical. CAS: 868540-17-4. Formula: C40H57N5O7. MW: 719.9. Synthetic. Potent and irreversible second-generation peptide epoxyketone class proteasome inhibitor. Synthetic analog of the microbial product epoxomcin. Targets the chymotrypsin-like beta5 subunit of the constitutive 20S proteasome (IC50=5.2nM)...
| Keywords: | (alphaS)-alpha-[[2-(4-Morpholinyl)acetyl]amino]benzenebutanoyl-L-leucyl-N-[(1S)-3-methyl-1-[[(2R)-2-methyl-2-oxiranyl]carb... |
| Application: | Proteasome inhibitor |
| CAS | 868540-17-4 |
| MW: | 719,9 D |
From 33.00€
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Carfilzomib, Free Base (Kyprolis, PR-171, CAS...
Item number: LC-C-3022_100mg
Soluble in DMSO
| Keywords: | PR-171,... |
| Application: | Proteasome PSMB5 inhibitor |
| CAS | 868540-17-4 |
| MW: | 719,91 D |
From 83.00€
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