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CMPD101
Item number: Cay26808-1
CMPD101 is an inhibitor of G protein-coupled receptor kinase 2 (GRK2) and GRK3 (IC50s = 18 and 5.4 nM, respectively). It is selective for GRK2 and GRK3 over GRK1, GRK5, GRK6, and GRK7 (IC50s = 3,100, 2,300, >30,000, and 25,000 nM, respectively), as well as Rho-associated kinase 2 (ROCK2) and PKCalpha (IC50s = 1,400...
| Keywords: | 3-[[[4-methyl-5-(4-pyridinyl)-4H-1,2,4-triazol-3-yl]methyl]amino]-N-[[2-(trifluoromethyl)phenyl]methyl]-benzamide |
| Application: | GRK2 inhibitor, GRK3 inhibitor |
| CAS | 865608-11-3 |
| MW: | 466.5 D |
From 50.00€
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CMPD101
Item number: TGM-T14989-1mg
Description: CMPD101 is a membrane-permeable small-molecule inhibitor of GRK2/3 (IC50: 18 nM and 5.4 nM). Which can be used for the study of heart failure. CMPD101 exhibits less selectively against GRK1, GRK5, ROCK-2 and PKCalpha with IC50s of 3.1 µM , 2.3 µM, 1.4 µM and 8.1 µM, respectively. Target: PKC, ROCK,...
| Application: | GRK2 inhibitor, GRK3 inhibitor |
| CAS | 865608-11-3 |
| MW: | 466.46 D |
From 40.00€
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