2 products were found matching "861238-35-9"!
No results were found for the filter!
DG-041
Item number: Cay13234-10
DG-041 is an antagonist of the prostaglandin E2 (PGE2, Cay-14010) receptor subtype EP3 (IC50 = 8.1 nM in a calcium mobilization assay). It is selective for EP3 over DP1, EP1, and TP receptors (IC50s = 131, 486, and 742 nM, respectively, in calcium mobilization assays) as well as EP2, EP4, IP, FP, and DP2/CRTH2...
| Keywords: | (2E)-3-[1-[(2,4-dichlorophenyl)methyl]-5-fluoro-3-methyl-1H-indol-7-yl]-N-[(4,5-dichloro-2-thienyl)sulfonyl]-2-propenamide |
| Application: | EP3 receptor antagonist |
| CAS | 861238-35-9 |
| MW: | 592.3 D |
From 126.00€
*
DG-041
Item number: TGM-T15108-100mg
Description: DG-041 is an antagonist of high affinity EP3 receptor (IC50s: 4.6 nM and 8.1 nM in the binding and FLIPR assay, respectively ). DG-041 inhibits PGE2 facilitation of platelet aggregation and it also crosses the blood-brain barrier. Target: Prostaglandin Receptor. Smiles:...
| Application: | EP3 receptor antagonist |
| CAS | 861238-35-9 |
| MW: | 592.32 D |
From 41.00€
*
