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Cariprazine
Item number: Cay31446-1
Cariprazine is an atypical antipsychotic. It binds to dopamine D2L, D2S, and D3 receptors, the serotonin (5-HT) receptor subtypes 5-HT1A, 5-HT2A, and 5-HT2B, and histamine H1 and sigma-1 (sigma1) receptors (Kis = 0.085-23.44 nM). Cariprazine is an antagonist of dopamine D2 and D3 receptors (Kbs = 0.759 and 0.316 nM,...
| Keywords: | RGH-188, N'-[trans-4-[2-[4-(2,3-dichlorophenyl)-1-piperazinyl]ethyl]cyclohexyl]-N,N-dimethyl-urea |
| Application: | Atypical antipsychotic, dopamine receptor partial agonist, serotonin receptor partial (ant)agonist |
| CAS | 839712-12-8 |
| MW: | 427.4 D |
From 49.00€
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Cariprazine
Item number: TGM-T4577-100mg
Description: Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (Ki=2.6 nM). Target: Dopamine Receptor, 5-HT Receptor. Smiles:...
| Keywords: | RGH-188 |
| Application: | Targets dopamine receptor D2 (DRD2) |
| CAS | 839712-12-8 |
| MW: | 427.41 D |
From 45.00€
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