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CID 16020046
Item number: TGM-T4478-100mg
Description: CID 16020046 (C390-0219) is a selective GPR55 antagonist, inhibiting GPR55 constitutive activity with IC50 of 0.15 µM in yeast. Target: Cannabinoid Receptor. Smiles: Cc1ccc(cc1)-c1n[nH]c2C(=O)N(C(c12)c1cccc(O)c1)c1ccc(cc1)C(O)=O. References: Kargl J, et al. A selective antagonist reveals a potential...
| Keywords: | C390-0219 |
| Application: | GPR55 inverse agonist |
| CAS | 834903-43-4 |
| MW: | 425.44 D |
From 34.00€
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CID-16020046
Item number: Cay15247-1
CID-16020046 is a GPR55 inverse agonist that antagonizes GPR55 constitutive activity with an IC50 value of 15 µM. It inhibits GPR55-mediated ERK1/2 phosphorylation, LPI-induced Ca2+ signaling (IC50 = 0.21 µM in HEK-GPR55 cells), and GPR55-mediated transcription factor activation. It does not affect ERK1/2...
| Keywords: | 4-[4,6-dihydro-4-(3-hydroxyphenyl)-3-(4-methylphenyl)-6-oxopyrrolo[3,4-c]pyrazol-5(1H)-yl]-benzoic acid |
| Application: | GPR55 inverse agonist |
| CAS | 834903-43-4 |
| MW: | 425.4 D |
From 49.00€
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