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PD 0332991 (hydrochloride)
PD 0332991 (hydrochloride)

Item number: Cay16273-1

PD 0332991 is an orally active, selective inhibitor of the cyclin D kinases Cdk4 (IC50 = 11 nM) and Cdk6 (IC50= 16 nM) with no activity against a panel of 36 additional protein kinases. It has been reported to have antiproliferative activity against retinoblastoma-positive tumor cells, blocking retinoblastoma...
Keywords: Palbociclib, 6-acetyl-8-cyclopentyl-5-methyl-2-[[5-(1-piperazinyl)-2-pyridinyl]amino]-pyrido[2,3-d]pyrimidin-7(8H)-one,...
Application: Cyclin-dependent kinase 4/6 (CDK4/6) inhibitor
CAS 827022-32-2
MW: 484 D
From 50.00€ *
Review
Palbociclib Hydrochloride
Palbociclib Hydrochloride

Item number: LKT-P0244.5

Palbociclib, also known as PD0332991, is an orally available pyridopyrimidine-derived cyclin-dependent kinase (CDK) inhibitor with potential antineoplastic activity. PD-0332991 selectively inhibits cyclin-dependent kinases (particularly Cdk4/cyclin D1 kinase), which may inhibit retinoblastoma (Rb) protein...
Keywords: PD-033291, PD0332991,...
Application: Cdk4 / Cdk6 inhibitor
CAS 827022-32-2
MW: 484 D
From 60.00€ *
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Palbociclib, Hydrochloride Salt (Ibrance, PD-0332991, PD 332991, CAS 827022-32-2), >99%
Palbociclib, Hydrochloride Salt (Ibrance, PD-0332991, PD...

Item number: LC-P-7788_100mg

Soluble in DMSO
Keywords: Palbociclib, 6-acetyl-8-cyclopentyl-5-methyl-2-[[5-(1-piperazinyl)-2-pyridinyl]amino]-pyrido[2,3-d]pyrimidin-7(8H)-one,...
Application: Cyclin-dependent kinase 4/6 (CDK4/6) inhibitor
CAS 827022-32-2
MW: 483,99 D
From 83.00€ *
Review