2 products were found matching "58-46-8"!

No results were found for the filter!
Tetrabenazine
Tetrabenazine

Item number: Cay20380-10

Tetrabenazine is an inhibitor of vesicular monoamine transporter 2 (VMAT2) that is selective over VMAT1 (Kis = 97 and >20,000 nM, respectively, in a serotonin uptake assay). It dose-dependently reduces levels of the monoamines norepinephrine (Cay-16673), dopamine (Cay-21992), and serotonin (5-HT, Cay-14332) in rat...
Keywords: NSC 169886, NSC 172187, Ro 1-9569, TBZ,...
Application: Neuroleptic, catecholamine uptake inhibitor
CAS 58-46-8
MW: 317.4 D
From 49.00€ *
Review
Tetrabenazine
Tetrabenazine

Item number: TGM-T0719-100mg

Description: Tetrabenazine (Ro 1-9569) is a former antipsychotic drug used to treat various movement disorders. It inhibits neurotransmitter uptake into adrenergic storage vesicles and serves as a high-affinity label for the vesicle transport system. Target: Monoamine Transporter, Dopamine Receptor, Others....
Keywords: Ro 1-9569, Xenazine
CAS 58-46-8
MW: 317.42 D
From 30.00€ *
Review