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BI-D1870
Item number: TGM-T6171-100mg
Description: BI-D1870 is a cell-permeable, ATP-competitive inhibitor of ribosomal S6 kinases (RSKs, IC50s: 31/24/18/15 nM for RSK1/2/3/4). Target: S6 Kinase, Autophagy. Smiles: CC(C)CCN1C(C)C(=O)N(C)c2cnc(Nc3cc(F)c(O)c(F)c3)nc12. References: Sapkota GP, et al. BI-D1870 is a specific inhibitor of the p90 RSK...
| Application: | RSK1/2/3/4 inhibitor |
| CAS | 501437-28-1 |
| MW: | 391.42 D |
From 48.00€
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BI-D1870
Item number: Cay15264-1
The 90 kDa ribosomal S6 kinases (RSKs) are a group of serine/threonine kinases involved in diverse cellular processes, including growth, survival, and motility. BI-D1870 is a cell permeable, ATP-competitive inhibitor of the four vertebrate isoforms of RSK, RSK1-4 (IC50s = 31, 24, 18, and 15 nM, respectively). At 100...
| Keywords: | 2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7,8-dihydro-5,7-dimethyl-8-(3-methylbutyl)-6(5H)-pteridinone |
| Application: | RSK1/2/3/4 inhibitor |
| CAS | 501437-28-1 |
| MW: | 391.4 D |
From 77.00€
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BI-D1870
Item number: SYN-1020-M001
Soluble in DMSO. Slightly soluble (<1mg/ml) in ethanol. BI-D1870 is a small molecule, specific inhibitor of p90 RSK (ribosomal S6 kinase) isoforms RSK1, RSK2, RSK3 and RSK4, both in vitro and in vivo, with IC(50)s are 31nM, 24nM, 18nM, 15nM, respectively. It shows a 10- to 100-fold selectivity for RSK over MST2,...
| Keywords: | BID1870 |
| Application: | RPS6KA inhibitor |
| CAS | 501437-28-1 |
| MW: | 391,4 D |
From 139.00€
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