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C646
Item number: Cay10549-1
C646 is an inhibitor of the histone acetyltransferase p300 (IC50 = 1.6 µM). It competitively (versus acetyl-CoA) binds p300 (Ki = 400 nM) and does not inhibit several other acetyltransferases. The action of C646 appears to be irreversible through covalent modification of the enzyme target. It blocks the growth of...
| Keywords: | 4-[4-[[5-(4,5-dimethyl-2-nitrophenyl)-2-furanyl]methylene]-4,5-dihydro-3-methyl-5-oxo-1H-pyra-zol-1-yl]-benzoic acid |
| Application: | Histone acetyltransferase p300 inhibitor |
| CAS | 328968-36-1 |
| MW: | 445.4 D |
From 50.00€
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C646
Item number: AG-CR1-3508-M001
Reversible cell permeable p300/CBP histone acetyltransferase (HAT) inhibitor. Specific inhibition to p300 (86% ) compared to N-acetyltransferase, PCAF, GCN5, Rtt109, Sas or MOZ histone acetyltransferases (<10% ). Cell growth inhibitor in melanoma and non-small-cell-lung (NSCL) human cancer cell lines.
| Keywords: | (E)-4-(4-((5-(4,5-Dimethyl-2-nitrophenyl)furan-2-yl)-methylene)-3-methyl-5-oxo-4,5-dihydro-1H-pyrazol-1-yl)benzoic acid |
| Application: | H2S donor |
| CAS | 328968-36-1 |
| MW: | 445,4 D |
From 39.00€
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