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AL 082D06
AL 082D06

Item number: Cay23455-1

AL 082D06 is a non-steroidal antagonist of the glucocorticoid receptor (GR, Ki = 210 nM, EC50 = 0.3 nM in a luciferase assay). It is selective for GR over the androgen, progesterone, mineralocorticoid, and estrogen receptors with Ki values greater than 4, 3, 3, and 10 µM, respectively. AL 082D06 inhibits...
Keywords: 4,4'-[(2-chloro-5-nitrophenyl)methylene]bis[N,N-dimethyl]-benzenamine
Application: Glucocorticoid receptor antagonist
CAS 256925-03-8
MW: 409.9 D
From 67.00€ *
Review
AL 082D06
AL 082D06

Item number: TGM-T1749-100mg

Description: AL 082D06 (D-06), a selective nonsteroidal glucocorticoid receptor (GR) antagonist (Ki: 210 nM), exhibits outstanding selectivity against AR, ER, MR and PR(Ki > 10 uM). Target: Glucocorticoid Receptor. Smiles: CN(C)c1ccc(cc1)C(c1ccc(cc1)N(C)C)c1cc(ccc1Cl)[N+]([O-])=O. References: Miner JN, et al. A...
Keywords: D-06, AL082D06
Application: Glucocorticoid receptor antagonist
CAS 256925-03-8
MW: 409.91 D
From 41.00€ *
Review