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Spastazoline
Item number: Cay43034-10
Spastazoline is an inhibitor of spastin (IC50 = 99 nM for the human enzyme). It is selective for spastin over a panel of 64 kinases but does inhibit tropomyosin-related kinase A (TrkA) by 65% at 2 µM. Spastazoline (10 µM) increases the number of cells with intracellular bridges during cell division, indicating...
| Keywords: | N-[5-(1,1-dimethylethyl)-1H-pyrazol-3-yl]-2-[(3R)-3-(1-methylethyl)-1-piperazinyl]-7H-pyrrolo[2,3-d]pyrimidin-4-amine |
| Application: | Spastin inhibitor |
| CAS | 2351882-11-4 |
| MW: | 382.52 D |
From 212.00€
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Spastazoline
Item number: TGM-T8513-100mg
Description: Spastazoline is a potent and selective inhibitor of spastin(Human spastin with IC50 of 99 nM ). Target: Others. Smiles: CC(C)[C@@H]1CN(CCN1)c1nc(Nc2cc([nH]n2)C(C)(C)C)c2cc[nH]c2n1. References: Cupido T, et al. Designing a chemical inhibitor for the AAA protein spastin using active site mutations. Nat...
| CAS | 2351882-11-4 |
| MW: | 382.51 D |
From 30.00€
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