2 products were found matching "2172870-89-0"!

No results were found for the filter!
Paltusotine
Paltusotine

Item number: TGM-T9692-100mg

Description: Paltusotine is a nonpeptide, small molecule somatostatin type 2 (SST2) receptor agonist with high oral bioavailability. Paltusotine maintains GH and IGF-1 levels in acromegaly patients. Target: Somatostatin. Smiles: NC1CCN(CC1)c1c(cnc2ccc(cc12)-c1cccc(C#N)c1O)-c1cc(F)cc(F)c1
Application: Targets somatostatin receptor 2 (SSTR2)
CAS 2172870-89-0
MW: 456.49 D
From 168.00€ *
Review
Paltusotine
Paltusotine

Item number: Cay42041-10

An SST2 agonist, selectively inhibits cAMP production in cells expressing SST2 over cells expressing SST1, SST3, SST4, or SST5 (EC50s = 25, >1,000, >1,000, >1,000, and >1,000 nM, respectively), reduces GHRH-stimulated growth hormone release in rats at 3, 10, and 30 mg/kg, reduces plasma levels of IGF-1 in beagle...
Keywords: CRN00808, 3-[4-(4-amino-1-piperidinyl)-3-(3,5-difluorophenyl)-6-quinolinyl]-2-hydroxy-benzonitrile
Application: SST2 agonist
CAS 2172870-89-0
MW: 456.5 D
From 421.00€ *
Review