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Item number: TGM-TQ0012-100mg

Description: AZ3451 is an allosteric antagonist of protease-activated receptor-2 (PAR2, IC50: 23 nM). Target: Protease-activated Receptor. Smiles: C[C@@H](C1CCCCC1)n1c(nc2cc(ccc12)C(=O)Nc1ccc(cc1)C#N)-c1cc2OCOc2cc1Br. References: Cheng RKY, et al. Structural insight into allosteric modulation of protease-activated...

Application:	Allosteric PAR2 antagonist
CAS	2100284-59-9
MW:	571.46 D

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AZ3451

Item number: Cay29671-1

AZ3451 is an allosteric antagonist of proteinase-activated receptor 2 (PAR2) that inhibits calcium mobilization by wild-type and 10 mutant forms of PAR2 induced by the PAR2 ligand SLIGRL in a FLIPR assay (IC50s = 23 and 12-780 nM, respectively). It is selective for PAR2 over PAR4 and PAR1 (IC50s = 50,000 nM,...

Keywords:	2-(6-bromo-1,3-benzodioxol-5-yl)-N-(4-cyanophenyl)-1-[(1S)-1-cyclohexylethyl]-1H-benzimidazole-5-carboxamide
Application:	Allosteric PAR2 antagonist
CAS	2100284-59-9
MW:	571.5 D

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