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Bilastine
Bilastine

Item number: TGM-T4250-100mg

Description: Bilastine (Bilaxten) is a novel new-generation antihistamine that is highly selective for the H1 histamine receptor, has a rapid onset and prolonged duration of action. Target: Histamine Receptor. Smiles: CCOCCn1c(nc2ccccc12)C1CCN(CCc2ccc(cc2)C(C)(C)C(O)=O)CC1. References: Wolthers OD.Bilastine: a new...
Keywords: Bilaxten
Application: Targets histamine receptor H1 (HRH1)
CAS 202189-78-4
MW: 463.61 D
From 40.00€ *
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Bilastine
Bilastine

Item number: Cay28375-25

Bilastine is a histamine H1 receptor antagonist (IC50 = 180 nM). It is selective for the histamine H1 receptor in a panel of 30 receptors in vitro at 100 µM. Bilastine prevents microvascular extravasation (ED50 = 185 µg/kg, i.v.), bronchospasm (ED50 = 4.6 µg/kg, i.v.), and systemic anaphylaxis (ED50 = 0.2 µg/kg,...
Keywords: F-96221-BM1, 4-[2-[4-[1-(2-ethoxyethyl)-1H-benzimidazol-2-yl]-1-piperidinyl]ethyl]-alpha,alpha-dimethyl-benzeneacetic acid
Application: Histamine H1 receptor antagonist
CAS 202189-78-4
MW: 463.6 D
From 61.00€ *
Review