2 products were found matching "199864-86-3"!

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Item number: Cay23451-1

RS 127445 is an orally bioavailable and potent antagonist of the serotonin (5-HT) receptor subtype 5-HT2B (Ki = 0.32 nM). It is selective for 5-HT2B over other 5-HT receptor subtypes (Ki = >3 µM for 5-HT1A, 5-HT1B, 5-HT2A, 5-HT2C, 5-HT3, 5-HT5, and 5-HT6). RS 127445 reduces contraction of rat isolated stomach fundus...

Keywords:	4-(4-fluoro-1-naphthalenyl)-6-(1-methylethyl)-2-pyrimidinamine
Application:	Serotonin (5-HT) receptor subtype 5-HT2B antagonist
CAS	199864-86-3
MW:	317.8 D

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RS-127445 hydrochloride

Item number: TGM-T7519-100mg

Description: RS-127445 hydrochloride (MT 500) is a selective, high affinity, orally bioavailable 5-HT2B receptor antagonist(pKi : 9.5). Target: 5-HT Receptor. Smiles: Cl.CC(C)c1cc(nc(N)n1)-c1ccc(F)c2ccccc12. References: Bonhaus D W , Flippin L A , Greenhouse R J , et al. RS-127445: a selective, high affinity, orally...

Keywords:	RS 127445 HCL , MT 500 HCL
Application:	Serotonin (5-HT) receptor subtype 5-HT2B antagonist
CAS	199864-86-3
MW:	317.79 D

From 30.00€ *

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