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PZM21
Item number: Cay20576-5
PZM21 is a µ-opioid receptor agonist (Ki = 1.1 nM). It is selective for µ- over kappa- and delta-opioid receptors (Kis = 18 and 506 nM, respectively). PZM21 induces Gi/o signaling (EC50 = 4.6 nM in HEK293T cells expressing human receptors) but has no detectable activity in a beta-arrestin2 recruitment assay. In...
| Keywords: | N-[(2S)-2-(dimethylamino)-3-(4-hydroxyphenyl)propyl]-N'-[(1S)-1-methyl-2-(3-thienyl)ethyl]-urea |
| Application: | ?-opioid receptor agonist |
| CAS | 1997387-43-5 |
| MW: | 361.5 D |
From 50.00€
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PZM21
Item number: TGM-T4386-100mg
Description: PZM21 is an effective and selective µ opioid receptor agonist (EC50: 1.8 nM). Target: Opioid Receptor. Smiles: C[C@@H](Cc1ccsc1)NC(=O)NC[C@H](Cc1ccc(O)cc1)N(C)C. References: Manglik A, et al. Structure-based discovery of opioid analgesics with reduced side effects. Nature. 2016 Sep 8,537(7619):185-190.
| Application: | ?-opioid receptor agonist |
| CAS | 1997387-43-5 |
| MW: | 361.5 D |
From 38.00€
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