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Valemetostat
Item number: Cay31674-500
Valemetostat is a dual inhibitor of enhancer of zeste homolog 1 (EZH1) and EZH2. It inhibits polycomb repressive complex 2 (PRC2) containing EZH1 or EZH2 as the catalytic subunit in cell-free assays (IC50s = 8.4 and 2.5 nM, respectively). Valemetostat inhibits trimethylation of histone H3 lysine 27 in HCT116 cells...
| Keywords: | (R)-OR-S2, DS-3201b,... |
| Application: | Antineoplastic, histone methyltransferase (EZH1/EZH2) inhibitor |
| CAS | 1809336-39-7 |
| MW: | 488 D |
From 80.00€
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Valemetostat
Item number: TGM-T13279L-100mg
Description: Valemetostat (DS-3201) is a first-in-class EZH1/2 dual inhibitor. Target: Histone Methyltransferase. Smiles: [H][C@@]1(CC[C@@H](CC1)N(C)C)[C@@]1(C)Oc2c(O1)c(C)c(cc2Cl)C(=O)NCc1c(C)cc(C)[nH]c1=O. References: Daiichi Sankyo's EZH1/2 Dual Inhibitor Valemetostat (DS-3201) Receives SAKIGAKE Designation for...
| Keywords: | DS-3201 |
| Application: | Antineoplastic, histone methyltransferase inhibitor |
| CAS | 1809336-39-7 |
| MW: | 488.02 D |
From 90.00€
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