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PLX51107
Item number: TGM-TQ0253-100mg
Description: PLX51107 is a potent and selective BET inhibitor with Kds of 1.6, 2.1, 1.7, and 5 nM for BRD2-BD1, BRD3-BD1, BRD4-BD1, and BRDT-BD1, respectively. Target: Epigenetic Reader Domain. Smiles: C[C@@H](c1ccccn1)n1cc(-c2ccc(cc2)C(O)=O)c2ncc(cc12)-c1c(C)noc1C. References: Ozer HG, et al. BRD4 Profiling...
| Application: | BET family protein inhibitor |
| CAS | 1627929-55-8 |
| MW: | 438.48 D |
From 52.00€
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PLX51107
Item number: Cay30742-5
PLX51107 is a bromodomain and extra terminal domain (BET) family protein inhibitor. It binds to bromodomain 1 (BD1) in bromodomain-containing protein 2 (BRD2), BRD3, BRD4, and BRDT (Kds = 1.6, 2.1, 1.7, and 5 nM, respectively), as well as BD2 (Kds = 5.9, 6.2, 6.1, and 120 nM, respectively). It also binds to the...
| Keywords: | 4-[6-(3,5-dimethyl-4-isoxazolyl)-1-[(1S)-1-(2-pyridinyl)ethyl]-1H-pyrrolo[3,2-b]pyridin-3-yl]-benzoic acid |
| Application: | BET family protein inhibitor |
| CAS | 1627929-55-8 |
| MW: | 438.5 D |
From 78.00€
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