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(R)-PFI-2 (hydrochloride)
Item number: Cay14678-1
SET domain-containing protein 7/9 (SET7/9) is a histone methyltransferase that monomethylates lysine 4 of histone H3, which generates a specific tag for epigenetic transcriptional activation. It plays a role in the transcriptional activation of tumor suppressor p53 in response to DNA damage as well as the...
| Keywords: | (-)-PFI-2,... |
| Application: | Cell-permeable SET7/9 inhibitor |
| CAS | 1627607-87-7 |
| MW: | 536 D |
From 40.00€
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PFI-2 hydrochloride
Item number: TGM-T4583-100mg
Description: PFI-2 hydrochloride ((R)-PFI-2 hydrochloride) is a potent, highly selective, and cell-active inhibitor of the methyltransferase activity of SETD7 (IC50: 2 nM), 500 fold active than (S)-PFI-2. Target: Histone Methyltransferase. Smiles: Cl.Fc1cc(cc2CCNCc12)S(=O)(=O)N[C@H](Cc1cccc(c1)C(F)(F)F)C(=O)N1CCCC1....
| Keywords: | (R)-PFI-2 hydrochloride, PFI-2 HCl |
| Application: | Cell-permeable SET7/9 inhibitor |
| CAS | 1627607-87-7 |
| MW: | 535.98 D |
From 33.00€
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