2 products were found matching "1621175-65-2"!
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TC-G-1008
Item number: TGM-T4648-100mg
Description: TC-G-1008 (GPR39-C3) is a zinc receptor agonist with EC50 values of 0.4 nM for rat GPR39 and 0.8 nM for human GPR39. Target: GHSR. Smiles: CNc1nc(NCc2ccc(NS(C)(=O)=O)cc2Cl)cc(n1)-c1ccccn1. References: Peukert S, et al. Discovery of 2-Pyridylpyrimidines as the First Orally Bioavailable GPR39 Agonists....
| Keywords: | GPR39-C3 |
| Application: | GPR39 agonist |
| CAS | 1621175-65-2 |
| MW: | 418.9 D |
From 42.00€
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GPR39-C3
Item number: Cay25445-1
GPR39-C3 is a potent agonist of the orphan G protein-coupled receptor GPR39 with EC50 values of 0.8 and 0.4 nM for cAMP production in HEK293 cells expressing human and rat receptors, respectively. It is selective for GPR39 over a panel of kinases (IC50s = >10 µM), ghrelin and neurotensin-1 receptors (IC50s = >30...
| Keywords: | N-[3-chloro-4-[[[2-(methylamino)-6-(2-pyridinyl)-4-pyrimidinyl]amino]methyl]phenyl]-methanesulfonamide |
| Application: | GPR39 agonist |
| CAS | 1621175-65-2 |
| MW: | 418.9 D |
From 45.00€
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