3 products were found matching "1395084-25-9"!
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MS436
Item number: LKT-M7200.1
BRD4 inhibitor.
| Application: | BRD4 inhibitor |
| CAS | 1395084-25-9 |
| MW: | 383.43 D |
From 128.00€
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MS436
Item number: TGM-T1854-100mg
Description: MS436 is a selective, small-molecule inhibitor for the BRD4 bromodomains. Target: Epigenetic Reader Domain. Smiles: Cc1cc(\N=N\c2ccc(cc2)S(=O)(=O)Nc2ccccn2)c(N)cc1O. References: Zhang G, et al. J Med Chem. 2013, 56(22), 9251-9264.
| Application: | Bromodomain inhibitor, BRD4 inhibitor |
| CAS | 1395084-25-9 |
| MW: | 383.42 D |
From 36.00€
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MS-436
Item number: BPS-82061-1
MS-436, through a set of water-mediated interactions, exhibits low nanomolar affinity (estimated Ki of 30-50 nM) to BRD4 with preference for the first bromodomain over the second. MS-436 effectively blocks BRD4 transcriptional activity in lipopolysaccharide-induced production of both nitric oxide and IL-6 in mouse...
| Keywords: | MS436, MS 436, |
| Application: | Bromodomain inhibitor, BRD4 inhibitor |
| CAS | 1395084-25-9 |
| MW: | 383,4 D |
From 1,228.00€
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