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JD5037
Item number: Cay12053-1
JD5037 is an inverse agonist of peripheral cannabinoid 1 (CB1) receptors (Ki = 0.35 nM). It displays >700-fold selectivity for CB1 over CB2, >1,000-fold selectivity over a panel of 70 receptors, transporters, and ion channels, and low blood-brain barrier penetrance. JD5037 is orally bioavailable and reduces food...
| Keywords: | 2S-[[[(4S)-3-(4-chlorophenyl)-4,5-dihydro-4-phenyl-1H-pyrazol-1-yl][[(4-chlorophenyl)sulfonyl]amino]methylene]amino]-3-met... |
| Application: | CB1 receptor inverse agonist |
| CAS | 1392116-14-1 |
| MW: | 572.5 D |
From 38.00€
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JD-5037
Item number: TGM-T4453-100mg
Description: JD-5037 is a novel, peripherally restricted CB1R antagonist with an IC50 of 1.5 nM. Target: Cannabinoid Receptor. Smiles: CC(C)[C@H](\N=C(\NS(=O)(=O)c1ccc(Cl)cc1)N1C[C@@H](C(=N1)c1ccc(Cl)cc1)c1ccccc1)C(N)=O. References: Knani I,etal.Targeting the endocannabinoid/CB1 receptor system for treating obesity...
| Keywords: | JD 5037 |
| CAS | 1392116-14-1 |
| MW: | 572.51 D |
From 36.00€
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