2 products were found matching "1365888-06-7"!

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Item number: Cay29595-5

ARN810 is a selective estrogen receptor degrader (SERD) that binds to ERalpha and ERbeta (IC50s = 6.1 and 8.8 nM, respectively) and induces degradation of ERalpha in MCF-7 cells (EC50 = 0.7 nM). It inhibits ERalpha transcriptional activity induced by 17beta-estradiol (Cay-10006315) in a reporter assay and reduces...

Keywords:	GDC-0810, RG-6046, (2E)-3-[4-[(1E)-2-(2-chloro-4-fluorophenyl)-1-(1H-indazol-5-yl)-1-buten-1-yl]phenyl]-2-propenoic acid
Application:	Selective estrogen receptor degrader (SERD)
CAS	1365888-06-7
MW:	446.9 D

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Brilanestrant

Item number: TGM-T5118-100mg

Description: Brilanestrant (GDC-0810) is a selective estrogen receptor degrader (IC50: 0.7 nM). Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor. Smiles: CC\C(=C(\c1ccc(\C=C\C(O)=O)cc1)c1ccc2[nH]ncc2c1)c1ccc(F)cc1Cl. References: By Lai, et al. Identification of GDC-0810 (ARN-810), an Orally Bioavailable...

Keywords:	ARN-810, RG 6046, GDC-0810, GDC 0810, GDC0810
Application:	Antineoplastic, Estrogen receptor degrader
CAS	1365888-06-7
MW:	446.9 D

From 46.00€ *

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