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Lintitript
Lintitript

Item number: TGM-T15759-100mg

Description: Lintitript (SR 27897) is a selective CCK1 antagonist with an EC50 of 6 nM for CCK1 and 200 nM for CCK2, and a Ki value of 0.2 nM for CCK1. Target: cholecystokinin. Smiles: OC(=O)Cn1c(cc2ccccc12)C(=O)Nc1nc(cs1)-c1ccccc1Cl. References: Gully D, et al. Peripheral biological activity of SR 27897: a new...
Keywords: SR 27897
Application: Cholecystokinin-1 receptor antagonist
CAS 136381-85-6
MW: 411.86 D
From 117.00€ *
Review
SR 27897
SR 27897

Item number: Cay28511-10

SR 27897 is a nonpeptide cholecystokinin (CCK) receptor antagonist. It selectively binds to CCK1 receptors in rat pancreatic membranes (IC50 = 0.58 nM) over CCK2 receptors in guinea pig cortical membranes and gastrin receptors in guinea pig gastric gland suspensions (IC50s = 489 and 2,883 nM, respectively). SR 27897...
Keywords: Lintitript, 2-[[[4-(2-chlorophenyl)-2-thiazolyl]amino]carbonyl]-1H-indole-1-acetic acid
Application: Cholecystokinin-1 receptor antagonist
CAS 136381-85-6
MW: 411.9 D
From 161.00€ *
Review