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PF-3644022
Item number: TGM-T16501-100mg
Description: PF-3644022 is an effective, selective, and ATP-competitive MAPKAPK2 (MK2) inhibitor (IC50: 5.2 nM and a Ki of 3 nM). PF-3644022 potently inhibits TNFalpha production and has an anti-inflammatory effect. PF-3644022 also inhibits MK3 and p38 regulated/activated kinase (PRAK) (IC50s: 53 nM and 5.0 nM,...
| Application: | MAPK-activated protein kinase 2 (MK2, MAPKAPK2) inhibitor |
| CAS | 1276121-88-0 |
| MW: | 374.46 D |
From 31.00€
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PF-3644022
Item number: Cay19185-1
PF-3644022 is an inhibitor of MAPK-activated protein kinase 2 (MK2, IC50 = 5.2 nM). It is selective for MK2 over MK3, MAPK-interacting protein kinase 1 (MNK-1), MNK-2, p90 ribosomal S6 kinase 1 (MSK1), MSK2, and p90 ribosomal S6 kinases 1-4 (RSK1-4, IC50s = 53, 3,000, 148, >1,000, >1,000, and >1,000 nM,...
| Keywords: | (10R)-9,10,11,12-tetrahydro-10-methyl-3-(6-methyl-3-pyridinyl)-8H-[1,4]diazepino[5',6':4,5]thieno[3,2-f]quinolin-8-one |
| Application: | MAPK-activated protein kinase 2 (MK2, MAPKAPK2) inhibitor |
| CAS | 1276121-88-0 |
| MW: | 374.5 D |
From 49.00€
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