2 products were found matching "126766-32-3"!

No results were found for the filter!
GR89696 (fumarate)
GR89696 (fumarate)

Item number: Cay40145-10

GR89696 is a kappa-opioid receptor agonist. It inhibits twitch responses in isolated mouse vas deferens (IC50 = 0.12 nM), an effect that can be reversed by the kappa-opioid receptor antagonist norbinaltorphimine (nor-BNI). In vivo, GR89696 reduces acetylcholine-induced writhing in mice (ED50 = 0.0005 mg/kg). It...
Keywords: 4-[2-(3,4-dichlorophenyl)acetyl]-3-(1-pyrrolidinylmethyl)-1-piperazinecarboxylic acid, methyl ester, (2E)-2-butenedioate
Application: Kappa-opioid receptor agonist
CAS 126766-32-3
MW: 530.4 D
From 132.00€ *
Review
GR 89696 fumarate
GR 89696 fumarate

Item number: TGM-T22810-100mg

Description: GR 89696 fumarate is a highly selective kappa2 opioid receptor agonist (IC50 = 0.04nM) with anti-pruritchy, anti-injury and neuroprotective effects. Target: Opioid Receptor. Smiles: C(=C/C(O)=O)\C(O)=O.C(CC1=CC(Cl)=C(Cl)C=C1)(=O)N2C(CN3CCCC3)CN(C(OC)=O)CC2. References: A Barber, et al. Effects of...
CAS 126766-32-3
MW: 530.4 D
From 55.00€ *
Review