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Azasetron hydrochloride
Item number: TGM-T1528-100mg
Description: Azasetron hydrochloride (Y-25130 HCl) is a 5-HT3 receptor antagonist which is used as an anti-emetic. Target: 5-HT Receptor. Smiles: Cl.CN1C(=O)COc2c1cc(Cl)cc2C(=O)NC1CN2CCC1CC2. References: Katayama K, et al. Jpn J Pharmacol. 1997 Apr,73(4):357-60.
| Keywords: | Y-25130 hydrochloride, Y-25130 HCl, Azasetron HCl |
| Application: | Targets 5-hydroxytryptamine receptor 3 (HTR3) |
| CAS | 123040-16-4 |
| MW: | 386.27 D |
From 34.00€
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Azasetron (hydrochloride)
Item number: Cay28383-10
Azasetron is an orally bioavailable antagonist of the serotonin (5-HT) receptor subtype 5-HT3 (Ki = 2.9 nM). It is selective for 5-HT3 over 5-HT1A and 5-HT2 (IC50 = >10 µM for both), as well as dopamine D1 and D2 and alpha1- and alpha2-adrenergic receptors (IC50s = >10 µM), but it does bind to histamine H1 receptors...
| Keywords: | Y-25130, N-1-azabicyclo[2.2.2]oct-3-yl-6-chloro-3,4-dihydro-4-methyl-3-oxo-2H-1,4-benzoxazine-8-carboxamide,... |
| Application: | Serotonin receptor 5-HT3 antagonist |
| CAS | 123040-16-4 |
| MW: | 386.3 D |
From 133.00€
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