2 products were found matching "121584-18-7"!

No results were found for the filter!
PSC 833
PSC 833

Item number: Cay20391-1

PSC 833 is a non-immunosuppressant derivative of cyclosporine and potent multidrug-resistance (MDR) modulator. It restores sensitivity of MDR-P388 murine leukemia cells to cytostatic agents when used at concentrations of 70, 33, 45, 34, and 26 nM in combination with colchicine, vincristine (Cay-11764), daunorubicin...
Keywords: Valspodar, 6-[(2S,4R,6E)-4-methyl-2-(methylamino)-3-oxo-6-octenoic acid]-7-L-valine-cyclosporin A
Application: MDR modulator
CAS 121584-18-7
MW: 1214.6 D
From 53.00€ *
Review
Valspodar
Valspodar

Item number: TGM-T17216-10mg

Description: Valspodar (PSC 833), a specific P-glycoprotein inhibitor and MDR regulator, is commonly used as a chemical sensitizer in the study of advanced epithelial ovarian cancer. Target: P-gp. Smiles:...
Keywords: PSC 833
Application: Targets ATP-binding cassette, subfamily B (MDR/TAP), member 1 [EC:7.6.2.2] (ABCB1, CD243)
CAS 121584-18-7
MW: 1214.62 D
From 199.00€ *
Review