2 products were found matching "1014691-61-2"!

No results were found for the filter!
GSK0660
GSK0660

Item number: TGM-T2674-100mg

Description: GSK0660 is an antagonist and inverse agonist of PPARbeta/delta. Target: PPAR. Smiles: S(NC1=C(OC)C=C(NC2=CC=CC=C2)C=C1)(=O)(=O)C3=C(C(OC)=O)SC=C3. References: Savage SR, et al. Mol Vis. 2015 May 20,21:568-76.
Application: PPARdelta antagonist
CAS 1014691-61-2
MW: 418.49 D
From 40.00€ *
Review
GSK0660
GSK0660

Item number: Cay15272-5

GSK0660 is the first reported antagonist of PPARbeta/delta (IC50 = 155 nM) with no measurable affinity for PPARalpha or PPARgamma (IC50s > 10 µM). Because of the limited bioavailability of GSK0660, the related compound GSK3787 (Cay-15219) was developed as a selective PPARbeta/delta antagonist with more suitable...
Keywords: 3-[[[2-methoxy-4-(phenylamino)phenyl]amino]sulfonyl]-2-thiophenecarboxylic acid, methyl ester
Application: PPARdelta antagonist
CAS 1014691-61-2
MW: 418.5 D
From 133.00€ *
Review