TWIK-1/TREK-1-IN-1

Item number	Size	Delivery time	Price
TGM-T78868-25mg	25 mg	7 - 10 business days*	1,440.00€
TGM-T78868-50mg	50 mg	7 - 10 business days*	1,877.00€
TGM-T78868-100mg	100 mg	7 - 10 business days*	2,371.00€

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Description: Compound 2a, identified as TWIK-1/TREK-1-IN-1, acts as an inhibitor of the TREK-1, a... more

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Product information "TWIK-1/TREK-1-IN-1"

Description: Compound 2a, identified as TWIK-1/TREK-1-IN-1, acts as an inhibitor of the TREK-1, a two-pore domain potassium channel (K2p) that forms TREK-1 homodimers and TWIK-1/TREK-1 heterodimers, both significant for its role as an antidepressant target. Furthermore, TWIK-1/TREK-1-IN-3, a related compound, selectively inhibits these channels with IC50 values of 9.36 µM for TREK-1 homodimers and 14.6 µM for TWIK-1/TREK-1 heterodimers, demonstrating antidepressant-like effects [1]. Target: Potassium Channel

Supplier:	TargetMol
Supplier-Nr:	T78868

Properties

MW:	395.42 D
Formula:	C21H24F3NO3

Database Information

CAS :

1440532-30-8| Matching products

Handling & Safety

Storage:	-20°C
Shipping:	+20°C (International: +4°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

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