SGC-AAK1-1
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SGC-AAK1-1 is a dual inhibitor of AP2-associated protein kinase 1 (AAK1) and BMP2-inducible... more
Product information "SGC-AAK1-1"
SGC-AAK1-1 is a dual inhibitor of AP2-associated protein kinase 1 (AAK1) and BMP2-inducible kinase (BMP2K, Kis = 9.1 and 17 nM, respectively). It is selective for AAK1 and BMP2K over cyclin G-associated kinase (GAK) and serine/threonine kinase 16 (STK16, Kis = 1,700 and 270 nM, respectively). See the Structural Genomics Consortium (SGC) website for more information.Formal Name: N-[6-[3-[[(diethylamino)sulfonyl]amino]phenyl]-1H-indazol-3-yl]-cyclopropanecarboxamide. CAS Number: 2247894-32-0. Molecular Formula: C21H25N5O3S. Formula Weight: 427.5. Purity: >98%. Formulation: (Request formulation change), A solid. Solubility: DMSO: Sparingly Soluble: 1-10 mg/ml. SMILES: O=C(C1CC1)NC2=NNC3=C2C=CC(C4=CC(NS(=O)(N(CC)CC)=O)=CC=C4)=C3. InChi Code: InChI=1S/C21H25N5O3S/c1-3-26(4-2)30(28,29)25-17-7-5-6-15(12-17)16-10-11-18-19(13-16)23-24-20(18)22-21(27)14-8-9-14/h5-7,10-14,25H,3-4,8-9H2,1-2H3,(H2,22,23,24,27). InChi Key: UCBIQZUJJSVQHL-UHFFFAOYSA-N.
| Keywords: | N-[6-[3-[[(diethylamino)sulfonyl]amino]phenyl]-1H-indazol-3-yl]-cyclopropanecarboxamide |
| Supplier: | Cayman Chemical |
| Supplier-Nr: | 41118 |
Properties
| Application: | AAK1 / BMP2K dual inhibitor |
| MW: | 427.5 D |
| Formula: | C21H25N5O3S |
| Purity: | >98% |
| Format: | Solid |
Database Information
| CAS : | 2247894-32-0| Matching products |
| KEGG ID : | K08853 | Matching products |
Handling & Safety
| Storage: | -20°C |
| Shipping: | +20°C (International: -20°C) |
| Signal Word: | Warning |
| GHS Hazard Pictograms: |
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| H Phrases: | H302, H315, H319, H335 |
| P Phrases: | P261, P264, P270, P271, P280, P312, P321, P330, P301+P310, P302+P352, P304+P340, P305+P351+P338, P332+P313, P337+P313, P362+P364, P405, P403+P233, P501 |
Caution
Our products are for laboratory research use only: Not for administration to humans!
Our products are for laboratory research use only: Not for administration to humans!
Information about the product reference will follow.
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